Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50021196
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221986(CHEMBL392469 | H-Tyr-Pro-Phe-Phe-NH-CH2-CH2-NH Tic...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221986(CHEMBL392469 | H-Tyr-Pro-Phe-Phe-NH-CH2-CH2-NH Tic...)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]deltorphin 2 from delta-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataKi:  1.81nMAssay Description:Displacement of [3H]deltorphin 2 from delta-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataKi:  2.72nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221986(CHEMBL392469 | H-Tyr-Pro-Phe-Phe-NH-CH2-CH2-NH Tic...)
Affinity DataIC50:  25.1nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataIC50:  286nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed