Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50038509
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377387(CHEMBL260720)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | N-[3-(1H-imidazol-4-ylmethyl)-phenyl]eth...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377388(CHEMBL406316)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377398(Ro-115-1240 | CHEMBL257978)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377391(CHEMBL402388)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377391(CHEMBL402388)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377394(CHEMBL404566)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377406(CHEMBL255938)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238839(N-[2-Chloro-5-(1H-imidazol-2-yl)-5,6,7,8-tetrahydr...)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377389(CHEMBL256983)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377395(CHEMBL257800)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238834(4-(5-chloro-1-(1H-imidazol-2-yl)-2,3-dihydro-1H-in...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377399(CHEMBL260009)
Affinity DataEC50:  111nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377393(CHEMBL257977)
Affinity DataEC50:  142nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377390(CHEMBL256984)
Affinity DataEC50:  167nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377401(CHEMBL407308)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377386(CHEMBL406348)
Affinity DataEC50:  278nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377388(CHEMBL406316)
Affinity DataEC50:  319nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377397(CHEMBL402003)
Affinity DataEC50:  322nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377390(CHEMBL256984)
Affinity DataEC50:  327nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377389(CHEMBL256983)
Affinity DataEC50:  336nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377396(CHEMBL258007)
Affinity DataEC50:  364nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377396(CHEMBL258007)
Affinity DataEC50:  385nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377400(CHEMBL260116)
Affinity DataEC50:  426nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377408(CHEMBL255937)
Affinity DataEC50:  451nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238822(2-(2,3-dihydro-1H-inden-1-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50:  473nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377389(CHEMBL256983)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human cloned adrenergic alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377387(CHEMBL260720)
Affinity DataEC50:  634nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377396(CHEMBL258007)
Affinity DataEC50:  722nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377396(CHEMBL258007)
Affinity DataEC50:  791nMAssay Description:Agonist activity at human cloned adrenergic alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377387(CHEMBL260720)
Affinity DataEC50:  902nMAssay Description:Agonist activity at human cloned adrenergic alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377403(CHEMBL260575)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377404(CHEMBL260789)
Affinity DataEC50: >1.30E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377407(CHEMBL257801)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377401(CHEMBL407308)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377402(CHEMBL260576)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377393(CHEMBL257977)
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377393(CHEMBL257977)
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377392(CHEMBL257976)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377405(CHEMBL261304)
Affinity DataEC50: >2.90E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377400(CHEMBL260116)
Affinity DataEC50:  3.19E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377392(CHEMBL257976)
Affinity DataEC50:  4.34E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377402(CHEMBL260576)
Affinity DataEC50:  4.58E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377401(CHEMBL407308)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377403(CHEMBL260575)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377404(CHEMBL260789)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377405(CHEMBL261304)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha-2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377395(CHEMBL257800)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238822(2-(2,3-dihydro-1H-inden-1-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | N-[3-(1H-imidazol-4-ylmethyl)-phenyl]eth...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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