Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50031019
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305440(2-(3-(5-bromoisoindoline-2-carbonyl)-1-(2-chloroph...)
Affinity DataIC50: 0.220nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305415(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 0.410nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305422(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 0.490nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305403(N-(4-bromo-2-fluorobenzyl)-1-(2-chlorophenyl)-5-(4...)
Affinity DataIC50: 0.510nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305423(N-(azepan-1-yl)-1-(2-chlorophenyl)-5-(4-chlorophen...)
Affinity DataIC50: 0.520nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305404(N-(3-bromo-4-fluorobenzyl)-1-(2-chlorophenyl)-5-(4...)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305432(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-(4-f...)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305427(methyl 2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-...)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305396(N-(4-chlorobenzyl)-1-(2-chlorophenyl)-5-(4-chlorop...)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305397(N-(4-bromobenzyl)-1-(2-chlorophenyl)-5-(4-chloroph...)
Affinity DataIC50: 1.20nMAssay Description:Inverse agonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as stimulation of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305401(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305424(trans-1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cya...)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305417(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305419(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305395(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305438(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(7-(tri...)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305425(N-((1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl)-1-(2-chlo...)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305393(methyl 2-(1-(1-(2-chlorophenyl)-5-(4-chlorophenyl)...)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305398(N-(3-chlorobenzyl)-1-(2-chlorophenyl)-5-(4-chlorop...)
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305435(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-(4-f...)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305388(2-(3-(4-benzyl-4-hydroxypiperidine-1-carbonyl)-1-(...)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305433(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-(pyr...)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305399(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 4.10nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305400(1-(2-chlorophenyl)-5-(4-chlorophenyl)-N-(4-cyanobe...)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305405(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305439(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(5-fluo...)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305437(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(1,2,3,...)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305397(N-(4-bromobenzyl)-1-(2-chlorophenyl)-5-(4-chloroph...)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305418(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305402(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305428(methyl 2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-...)
Affinity DataIC50: 7.30nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305420(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305416(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 7.80nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305434(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(3-(4-f...)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305407(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305431(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-phen...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305409(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305414(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305413(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305391(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-(met...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305410(1-(2-chlorophenyl)-5-(4-chlorophenyl)-N-(2-chlorop...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305411(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305390(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-((R)-3-...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305436(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(2-(4-f...)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305389(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(2-(4-f...)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305426(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305412(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305408(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50305421(1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-(cyanometh...)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human recombinant CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-stimulated GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
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