Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50043297
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 75nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438825BDBM50438825(CHEMBL2413741)
Affinity DataIC50: 580nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438843BDBM50438843(CHEMBL2413743)
Affinity DataIC50: 610nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438830BDBM50438830(CHEMBL2413736)
Affinity DataIC50: 840nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438836BDBM50438836(CHEMBL2413560)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438838BDBM50438838(CHEMBL2413558)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438831BDBM50438831(CHEMBL2413735)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438830BDBM50438830(CHEMBL2413736)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438832BDBM50438832(CHEMBL2413734)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438836BDBM50438836(CHEMBL2413560)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438827BDBM50438827(CHEMBL2413739)
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438837BDBM50438837(CHEMBL2413559)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438831BDBM50438831(CHEMBL2413735)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438844BDBM50438844(CHEMBL2413742)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438844BDBM50438844(CHEMBL2413742)
Affinity DataIC50: 3.42E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438826BDBM50438826(CHEMBL2413740)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438838BDBM50438838(CHEMBL2413558)
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438841BDBM50438841(CHEMBL377740)
Affinity DataIC50: 4.59E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438834BDBM50438834(CHEMBL2413732)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438839BDBM50438839(CHEMBL2413745)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438833BDBM50438833(CHEMBL2413733)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438840BDBM50438840(CHEMBL2413746)
Affinity DataIC50: 5.87E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438832BDBM50438832(CHEMBL2413734)
Affinity DataIC50: 6.48E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438825BDBM50438825(CHEMBL2413741)
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438828BDBM50438828(CHEMBL2413738)
Affinity DataIC50: 8.52E+3nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438842BDBM50438842(CHEMBL2413744)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438840BDBM50438840(CHEMBL2413746)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438828BDBM50438828(CHEMBL2413738)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438839BDBM50438839(CHEMBL2413745)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438834BDBM50438834(CHEMBL2413732)
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438841BDBM50438841(CHEMBL377740)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438835BDBM50438835(CHEMBL2413561)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438837BDBM50438837(CHEMBL2413559)
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438835BDBM50438835(CHEMBL2413561)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438829BDBM50438829(CHEMBL2413737)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438833BDBM50438833(CHEMBL2413733)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438843BDBM50438843(CHEMBL2413743)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438827BDBM50438827(CHEMBL2413739)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438826BDBM50438826(CHEMBL2413740)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438842BDBM50438842(CHEMBL2413744)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Ege University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438829BDBM50438829(CHEMBL2413737)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide as substrate preincubated for 5 mins before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed