Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50006228
LigandChemical structure of BindingDB Monomer ID 124444BDBM124444(US8759532, 99)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 124447BDBM124447(US8759532, 103)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497975BDBM50497975(CHEMBL3319207)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50494199BDBM50494199(CHEMBL3086091)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50494193BDBM50494193(CHEMBL3086099)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497974BDBM50497974(CHEMBL3319209)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PDE2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed