Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50045708
LigandChemical structure of BindingDB Monomer ID 50077877BDBM50077877(CHEMBL3417042 | US9611229, 2)
Affinity DataKi:  5nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077891BDBM50077891(CHEMBL3417066 | US9611229, 12)
Affinity DataKi:  9nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077886BDBM50077886(CHEMBL3417058 | US9611229, 9)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50396335BDBM50396335(CHEMBL2170054)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077899BDBM50077899(CHEMBL3417052 | US9611229, 13)
Affinity DataKi:  12nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077905BDBM50077905(CHEMBL3417068 | US9611229, 33)
Affinity DataKi:  13nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50396352BDBM50396352(CHEMBL2170062)
Affinity DataKi:  17nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077892BDBM50077892(CHEMBL3417067 | US9611229, 15)
Affinity DataKi:  23nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077881BDBM50077881(CHEMBL3417047 | US9611229, 47)
Affinity DataKi:  31nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077878BDBM50077878(CHEMBL3417043 | US9611229, 3)
Affinity DataKi:  31nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077889BDBM50077889(CHEMBL3417061 | US9611229, 37)
Affinity DataKi:  33nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077888BDBM50077888(CHEMBL3417060 | US9611229, 18)
Affinity DataKi:  35nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077883BDBM50077883(CHEMBL3417054 | US9611229, 32)
Affinity DataKi:  36nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50396336BDBM50396336(CHEMBL2170053)
Affinity DataKi:  39nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077893BDBM50077893(CHEMBL3417069 | US9611229, 40)
Affinity DataKi:  46nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077882BDBM50077882(CHEMBL3417049 | US9611229, 5)
Affinity DataKi:  46nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077885BDBM50077885(CHEMBL3417057 | US9611229, 4)
Affinity DataKi:  49nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077887BDBM50077887(CHEMBL3417059 | US9611229, 17)
Affinity DataKi:  52nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077900BDBM50077900(CHEMBL3417053 | US9611229, 31)
Affinity DataKi:  56nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077880BDBM50077880(CHEMBL3417045 | US9611229, 46)
Affinity DataKi:  58nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077890BDBM50077890(CHEMBL3417063 | US9611229, 7)
Affinity DataKi:  61nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077879BDBM50077879(CHEMBL3417044 | US9611229, 39)
Affinity DataKi:  62nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077884BDBM50077884(CHEMBL3417055 | US9611229, 43)
Affinity DataKi:  70nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077869BDBM50077869(CHEMBL3417078 | US9611229, 6)
Affinity DataKi:  97nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077862BDBM50077862(CHEMBL3417071 | US9611229, 49)
Affinity DataKi:  99nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077894BDBM50077894(CHEMBL3417070 | US9611229, 41)
Affinity DataKi:  105nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077872BDBM50077872(CHEMBL3417081 | US9611229, 64)
Affinity DataKi:  111nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077895BDBM50077895(CHEMBL3417046 | US9611229, 48)
Affinity DataKi:  144nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077867BDBM50077867(CHEMBL3417076 | US9611229, 23)
Affinity DataKi:  194nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077870BDBM50077870(CHEMBL3417079 | US9611229, 65)
Affinity DataKi:  216nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077876BDBM50077876(CHEMBL3417085 | US9611229, 68)
Affinity DataKi:  241nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077896BDBM50077896(CHEMBL3417048 | US9611229, 50)
Affinity DataKi:  273nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077901BDBM50077901(CHEMBL3417056 | US9611229, 51)
Affinity DataKi:  275nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077873BDBM50077873(CHEMBL3417082)
Affinity DataKi:  388nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077871BDBM50077871(CHEMBL3417080)
Affinity DataKi:  451nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077874BDBM50077874(CHEMBL3417083)
Affinity DataKi:  459nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077866BDBM50077866(CHEMBL3417075)
Affinity DataKi:  508nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077862BDBM50077862(CHEMBL3417071 | US9611229, 49)
Affinity DataIC50: 600nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077903BDBM50077903(CHEMBL3417064)
Affinity DataKi:  662nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077863BDBM50077863(CHEMBL3417072)
Affinity DataKi:  701nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077897BDBM50077897(CHEMBL3417050)
Affinity DataKi:  781nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077865BDBM50077865(CHEMBL3417074)
Affinity DataKi:  818nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077904BDBM50077904(CHEMBL3417065)
Affinity DataKi:  878nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077868BDBM50077868(CHEMBL3417077)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077898BDBM50077898(CHEMBL3417051)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077875BDBM50077875(CHEMBL3417084)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077902BDBM50077902(CHEMBL3417062)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077877BDBM50077877(CHEMBL3417042 | US9611229, 2)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077881BDBM50077881(CHEMBL3417047 | US9611229, 47)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50077886BDBM50077886(CHEMBL3417058 | US9611229, 9)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
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