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Found 82 Enz. Inhib. hit(s) with all data for entry = 50006495
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50:  6nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50:  11nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500319(CHEMBL3746179)
Affinity DataIC50:  15nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500347(CHEMBL3747049)
Affinity DataIC50:  23nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50:  40nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163143(US9062026, Table III, Compound 71)
Affinity DataIC50:  43nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163134(US9062026, Table III, Compound 62)
Affinity DataIC50:  47nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163144(US9062026, Table III, Compound 72)
Affinity DataIC50:  68nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500321(CHEMBL3745888)
Affinity DataIC50:  71nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500323(CHEMBL3746353)
Affinity DataIC50:  76nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500318(CHEMBL3746650)
Affinity DataIC50:  95nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500339(CHEMBL3747498)
Affinity DataIC50:  98nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500316(CHEMBL3746000)
Affinity DataIC50:  144nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163082(US9062026, Table III, Compound 10)
Affinity DataIC50:  145nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500337(CHEMBL3747075)
Affinity DataIC50:  149nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163080(US9062026, Table III, Compound 8)
Affinity DataIC50:  152nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163136(US9062026, Table III, Compound 64 | US9062026, Tab...)
Affinity DataIC50:  153nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163092(US9062026, Table III, Compound 20)
Affinity DataIC50:  180nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163115(US9062026, Table III, Compound 43)
Affinity DataIC50:  192nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500320(CHEMBL3747639)
Affinity DataIC50:  215nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163098(US9062026, Table III, Compound 26)
Affinity DataIC50:  227nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163097(US9062026, Table III, Compound 25)
Affinity DataIC50:  233nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500312(CHEMBL3746787)
Affinity DataIC50:  248nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50:  250nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500335(CHEMBL3746988)
Affinity DataIC50:  304nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500309(CHEMBL3745805)
Affinity DataIC50:  342nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500307(CHEMBL3746833)
Affinity DataIC50:  367nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500331(CHEMBL3220939)
Affinity DataIC50:  370nMAssay Description:Inhibition of p97 ATPase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163139(US9062026, Table III, Compound 67)
Affinity DataIC50:  370nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500327(CHEMBL3746037)
Affinity DataIC50:  425nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163135(US9062026, Table III, Compound 63)
Affinity DataIC50:  445nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50:  490nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50:  500nMAssay Description:Inhibition of DNAPK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50:  500nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50:  580nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500332(CHEMBL3747140)
Affinity DataIC50:  632nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500315(CHEMBL3747371)
Affinity DataIC50:  648nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500306(CHEMBL3747138)
Affinity DataIC50:  651nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50:  680nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163145(US9062026, Table III, Compound 73)
Affinity DataIC50:  795nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500322(CHEMBL3746912)
Affinity DataIC50:  815nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163086(US9062026, Table III, Compound 14)
Affinity DataIC50:  907nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163106(US9062026, Table III, Compound 34)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500338(CHEMBL3747194)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500305(CHEMBL3747511)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163114(US9062026, Table III, Compound 42)
Affinity DataIC50:  3.13E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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