Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50012595
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120880(2-[(2-{2-[2-Amino-3-(3-hydroxy-phenyl)-propionylam...)
Affinity DataIC50: 10.2nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120878(2-[(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phe...)
Affinity DataIC50: 12.9nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120875(2-(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phen...)
Affinity DataIC50: 20.8nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120876(6-Amino-2-[(2-{5-guanidino-2-[2-guanidino-3-(3-hyd...)
Affinity DataIC50: 32.9nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120877(2-[(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methy...)
Affinity DataIC50: 45nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120879(2-[(2-{2-[2-Dimethylamino-3-(3-hydroxy-phenyl)-pro...)
Affinity DataIC50: 101nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120880(2-[(2-{2-[2-Amino-3-(3-hydroxy-phenyl)-propionylam...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120875(2-(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120879(2-[(2-{2-[2-Dimethylamino-3-(3-hydroxy-phenyl)-pro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120878(2-[(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120875(2-(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120874(2-(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120879(2-[(2-{2-[2-Dimethylamino-3-(3-hydroxy-phenyl)-pro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120876(6-Amino-2-[(2-{5-guanidino-2-[2-guanidino-3-(3-hyd...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120877(2-[(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120877(2-[(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120874(2-(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120874(2-(2-{5-Guanidino-2-[3-(3-hydroxy-phenyl)-2-methox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [3H]DAMGO in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120876(6-Amino-2-[(2-{5-guanidino-2-[2-guanidino-3-(3-hyd...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120878(2-[(2-{5-Guanidino-2-[2-guanidino-3-(3-hydroxy-phe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
Daiichi Fine Chemical

Curated by ChEMBL
LigandPNGBDBM50120880(2-[(2-{2-[2-Amino-3-(3-hydroxy-phenyl)-propionylam...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [3H]U-69593 in mouse spinal cordMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed