Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50012596
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558654BDBM50558654(CHEMBL4797972)
Affinity DataEC50:  98nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558648BDBM50558648(CHEMBL4778177)
Affinity DataEC50:  102nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558655BDBM50558655(CHEMBL4781319)
Affinity DataEC50:  119nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558649BDBM50558649(CHEMBL4778053)
Affinity DataEC50:  134nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10758BDBM10758(14C-phenylethylamine | 2-phenylethan-1-amine | CHE...)
Affinity DataEC50:  138nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558652BDBM50558652(CHEMBL4761622)
Affinity DataEC50:  158nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359505BDBM50359505(CHEMBL1182312)
Affinity DataEC50:  189nMAssay Description:Agonist activity at mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096963BDBM50096963(CHEMBL3580902)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558647BDBM50558647(CHEMBL4794080)
Affinity DataEC50:  440nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558650BDBM50558650(CHEMBL4800489)
Affinity DataEC50:  633nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558651BDBM50558651(CHEMBL4744061)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096964BDBM50096964(CHEMBL3580901)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558653BDBM50558653(CHEMBL4787435)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558640BDBM50558640(CHEMBL4763482)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558641BDBM50558641(CHEMBL4741294)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558642BDBM50558642(CHEMBL4741475)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558643BDBM50558643(CHEMBL4793672)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558644BDBM50558644(CHEMBL4781549)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558645BDBM50558645(CHEMBL4764889)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558646BDBM50558646(CHEMBL4797425)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR1 expressed in HEK293T cells assessed as induction of cAMP production by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed