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Found 43 Enz. Inhib. hit(s) with all data for entry = 5181
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  1.05nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  1.35nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  2.09nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
Affinity DataKi:  2.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  3.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  3.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  3.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  4.47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  6.76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  27.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  52.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
Affinity DataKi:  89.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  407nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed