Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 10537
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547776BDBM547776(Methyl (3R)-3-(((5R)-5-Oxido-2-(3-phenylazetidin-1...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547778BDBM547778(Methyl (3S)-3-(((5R)-2-(3-(4-Fluorophenoxy)azetidi...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547777BDBM547777(Methyl (3R)-3-(((5R)-2-(3-(4-Fluorophenoxy)azetidi...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547780BDBM547780((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-(4-flu...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547779BDBM547779((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-(4-flu...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547781BDBM547781((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-phenyl...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547784BDBM547784((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-(pyrid...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547783BDBM547783((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-(3-flu...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547785BDBM547785((R)-4-((1-Methylcyclobutyl)amino)-2-(3-(pyridin-2-...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547787BDBM547787((5R)—N-(1,1-Dioxothian-4-yl)-5-oxido-2-(3-phe...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547772BDBM547772((R)-2-(3-Phenylazetidin-1-yl)-4-((tetrahydro-2H-py...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547774BDBM547774((R)-2-(3-(4-Fluorophenoxy)azetidin-1-yl)-4-((tetra...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547773BDBM547773((R)-2-(3-Phenoxyazetidin-1-yl)-4-((tetrahydro-2H-p...)
Affinity DataIC50: 10nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547775BDBM547775(Methyl (3S)-3-(((5R)-5-oxido-2-(3-phenylazetidin-1...)
Affinity DataIC50: 30nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547782BDBM547782((R)-4-(Bicyclo[1.1.1]pentan-1-ylamino)-2-(3-(pyrid...)
Affinity DataIC50: 30nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D [538-740](Human)
Union Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 547786BDBM547786((R)-4-((1-Methylcyclobutyl)amino)-2-(3-(pyridin-3-...)
Affinity DataIC50: 30nMAssay Description:The human PDE4D catalytic domain (UniProt no. Q08499 [5380-L740]) was incubated with a mixture of non-labelled cAMP (cyclic adenosine monophosphate) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2022
Entry Details
US Patent