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Report error Found 2279 for UniProtKB: P08588
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50379086(CHEMBL2012522 | CHEMBL2012521 | LY-377604)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta1 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378919(CHEMBL2011218)
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378927(CHEMBL2011226)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378913(CHEMBL2011227)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50568740(CHEMBL4860528)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50601567(CHEMBL5206565)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50601551(CHEMBL5207281)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50601574(CHEMBL5201074)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378917(CHEMBL2011216)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50318983(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378925(CHEMBL2011224)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378916(CHEMBL2011215)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378914(CHEMBL2011213)
Affinity DataIC50: 0.110nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.114nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50126071((R)-1-((R)-3-Chloro-phenyl)-2-[2-(7-methoxy-1H-ind...)
Affinity DataEC50:  0.130nMAssay Description:Agonistic activity against human Beta-1 adrenergic receptor by measuring cAMP accumulation in CHO cells expressing beta3-ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50126076((R)-1-(3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at Homo sapiens (human) beta1 adrenoreceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378935(CHEMBL2011235)
Affinity DataIC50: 0.140nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378915(CHEMBL2011214)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378918(CHEMBL2011217)
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50098668(4-(3-tert-Butylamino-2-hydroxy-propoxy)-1,3-dihydr...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378926(CHEMBL2011225)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378928(CHEMBL2011228)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50241366((S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol (...)
Affinity DataKd:  0.380nMAssay Description:Binding affinity to beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity at human adrenergic beta-1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50328336(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-...)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at human recombinant adrenergic beta-1 receptor expressed in CHO cells assessed as cyclic AMP formation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50299900(5-hydroxy-8-(1-hydroxy-2-(2-methyl-1-o-tolylpropan...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human adrenergic beta 1 expressed in CHO-K1 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50578620(CHEMBL4868585)
Affinity DataEC50:  0.603nMAssay Description:Agonist activity at human beta1 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25747(4-[3-(tert-butylamino)-2-hydroxypropoxy]-2,3-dihyd...)
Affinity DataKd:  0.620nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50055260(CHEMBL3323658)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]iodo-(+/-)-cyanopindolol from human adrenergic beta1 receptor expressed in CHO cells after 3 hrs by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50299901(5-hydroxy-8-(1-hydroxy-2-(2-methyl-1-phenylpropan-...)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human adrenergic beta 1 expressed in CHO-K1 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataEC50:  0.813nMAssay Description:Partial agonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50578619(CHEMBL4862449)
Affinity DataEC50:  0.851nMAssay Description:Agonist activity at human beta1 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50027164(CHEMBL369346)
Affinity DataEC50:  0.900nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50324854(7-((R)-2-((1R,2R)-2-(benzyloxy)cyclopentylamino)-1...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50299890(5-hydroxy-8-(1-hydroxy-2-(1-(4-hydroxyphenyl)-2-me...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human adrenergic beta 1 expressed in CHO-K1 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50232757(CHEMBL4092412)
Affinity DataKd:  0.977nMAssay Description:Displacement of [3H](-)CGP12177 from human beta1-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/23/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50432704(CHEMBL2348218)
Affinity DataKd:  1nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50318987(1-(9H-carbazol-4-yloxy)-3-(4-(pyridin-3-ylmethyl)p...)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50378923(CHEMBL2011222)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  1nMAssay Description:Activity at human beta-1 adrenergic receptor expressed in CHO cells by stimulation of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article
PubMed
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