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TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataKd:  3.90E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataKd:  1.40E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  81nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  430nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13534(VX680 | N-[4-[[4-(4-methylpiperazino)-6-[(5-methyl...)
Affinity DataKd:  290nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2009
Entry Details
PCBioAssay
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50118239(uridine 5'-(trihydrogen diphosphate) | UDP | Uridi...)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human P2Y14 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50118239(uridine 5'-(trihydrogen diphosphate) | UDP | Uridi...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human P2Y14 expressed in rat C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50118239(uridine 5'-(trihydrogen diphosphate) | UDP | Uridi...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human P2Y14 expressed in rat CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50512416(CHEMBL4447162)
Affinity DataKd:  28nMAssay Description:Binding affinity to human P2Y14R stably expressed in CHO cells assessed as dissociation constant by Cheng-prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209658([({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydrop...)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209659(uridine 5'-[3-alpha-D-glucopyranosyl dihydrogen di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209661([({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydrop...)
Affinity DataEC50:  880nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209663(MRS-2670 | diphosphoric acid 1-alpha-D-glucopyrano...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209665(uridine 5'-[3-(alpha-D-glucopyranuronosyl) dihydro...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209664(diphosphoric acid 1-alpha-D-glucopyranosyl ester 2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209666(URIDINE-5'-DIPHOSPHATE-MANNOSE | CHEMBL227711)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209667(diphosphoric acid 1-alpha-D-glucopyranosuronic aci...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209669(MRS-2670 | diphosphoric acid 1-alpha-D-glucopyrano...)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209668(Galactose-Uridine-5'-Diphosphate | CHEMBL439009)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50197974(udp-N-acetyl-glucosamine)
Affinity DataEC50:  810nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50197974(udp-N-acetyl-glucosamine)
Affinity DataEC50:  810nMAssay Description:Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50638480(CHEMBL5557370)
Affinity DataKd:  0.110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50197974(udp-N-acetyl-glucosamine)
Affinity DataEC50:  4.38E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209659(uridine 5'-[3-alpha-D-glucopyranosyl dihydrogen di...)
Affinity DataEC50:  261nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209669(MRS-2670 | diphosphoric acid 1-alpha-D-glucopyrano...)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209663(MRS-2670 | diphosphoric acid 1-alpha-D-glucopyrano...)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304030(Diphosphoric Acid 1''-beta-D-[1'']Glucopyranosyl E...)
Affinity DataEC50:  588nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209666(URIDINE-5'-DIPHOSPHATE-MANNOSE | CHEMBL227711)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209668(Galactose-Uridine-5'-Diphosphate | CHEMBL439009)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304031(Diphosphoric Acid 1''-alpha-D-[1'']Fucopyranosyl E...)
Affinity DataEC50:  562nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304032(URIDINE-5'-DIPHOSPHATE-2-DEOXY-2-FLUORO-ALPHA-D-GL...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304033(Diphosphoric Acid 1''-alpha-D-[1''](3''-Fluoro-3''...)
Affinity DataEC50:  361nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304034(URIDINE-5'-DIPHOSPHATE-4-DEOXY-4-FLUORO-ALPHA-D-GA...)
Affinity DataEC50:  567nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304035(Diphosphoric Acid 1''-alpha-D-[1''](6''-Fluoro-6''...)
Affinity DataEC50:  905nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209665(uridine 5'-[3-(alpha-D-glucopyranuronosyl) dihydro...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304036(Diphosphoric acid 1''-alpha-D-[1''](glucuronic aci...)
Affinity DataEC50:  2.59E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304037({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydropyr...)
Affinity DataEC50:  496nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304038(Diphosphoric Acid 1''-alpha-D-[6'']Glucopyranosyl ...)
Affinity DataEC50:  373nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304039(Diphosphoric Acid 1''-alpha-D-[6'']Mannopyranosyl ...)
Affinity DataEC50:  658nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304040(Diphosphoric Acid 1''-alpha-D-[5'']Ribofuranosyl E...)
Affinity DataEC50:  238nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304041(Diphosphoric Acid 1''-alpha-D-[5'']Arabinofuranosy...)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50209661([({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydrop...)
Affinity DataEC50:  880nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304042(Diphosphoric Acid 1''-alpha-D-[1'']Fructofuranosyl...)
Affinity DataEC50:  323nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304043({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,4-tetrahydropyr...)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50304044([({[(2R,3R,4S,5S,6S)-6-[(2-{[(tert-butoxy)carbonyl...)
Affinity DataEC50:  951nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50197974(udp-N-acetyl-glucosamine)
Affinity DataEC50:  4.38E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50319129(CHEMBL1204010 | CHEMBL1084020 | N4-Methoxycytidine...)
Affinity DataEC50:  3.32E+3nMAssay Description:Agonist activity at human recombinant P2Y14 receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation proximi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50118239(uridine 5'-(trihydrogen diphosphate) | UDP | Uridi...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human recombinant P2Y14 receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation proximi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50319142(5-Iodouridine5'-Methylenediphosphate Triethylammon...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human recombinant P2Y14 receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation proximi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
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