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Report error Found 49 for UniProtKB: Q6GPI1
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520048BDBM50520048(CHEMBL4450993)
Affinity DataKi:  0.420nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520063BDBM50520063(CHEMBL4586444)
Affinity DataKi:  0.880nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520058BDBM50520058(CHEMBL4469390)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520064BDBM50520064(CHEMBL4590739)
Affinity DataKi:  11nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50541586BDBM50541586(CHEMBL4638245)
Affinity DataKi:  20nMAssay Description:Inhibition of human chymotrypsin by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 247411BDBM247411(US9453018, 353 | US10336754, Example 353 | US11053...)
Affinity DataKi:  35nMAssay Description:Binding affinity to human chymotrypsin assessed as inhibition constant using 3-Carbomethoxypropionyl-L-arginyl-Lprolyl-L-tyrosine p-Nitroaniline as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520051BDBM50520051(CHEMBL4592765)
Affinity DataKi:  150nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520049BDBM50520049(CHEMBL4560112)
Affinity DataKi:  330nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 162366BDBM162366(US9687479, 3 3-(5-[(5-chlorothiophen-2-yl)methyl]a...)
Affinity DataIC50: 380nMAssay Description:Inhibition of chymotrypsin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502655BDBM50502655(CHEMBL4560512)
Affinity DataKi:  463nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 163407BDBM163407(US9687479, 278 1-[(2-methoxyphenyl)carbonyl]-3-(py...)
Affinity DataIC50: 670nMAssay Description:Inhibition of chymotrypsin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520061BDBM50520061(CHEMBL4556207)
Affinity DataKi:  920nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520060BDBM50520060(CHEMBL4465306)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520050BDBM50520050(CHEMBL4457132)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548603BDBM50548603(CHEMBL4761275)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-Suc-Ala-Ala-Pro-Phe-pNA as chromogenic substrate incubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548594BDBM50548594(CHEMBL4776259)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-Suc-Ala-Ala-Pro-Phe-pNA as chromogenic substrate incubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520052BDBM50520052(CHEMBL4554739)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502656BDBM50502656(CHEMBL4455694)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502658BDBM50502658(CHEMBL4557877)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504368BDBM50504368(CHEMBL4435573)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibition of human chymotrypsin using S-2586 as substrate incubated for 15 mins followed by substrate addition and measured after 1 hr by chromogeni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533255BDBM50533255(CHEMBL4476255)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533255BDBM50533255(CHEMBL4476255)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50504369BDBM50504369(CHEMBL4439549)
Affinity DataKi:  1.63E+4nMAssay Description:Inhibition of human chymotrypsin using S-2586 as substrate incubated for 15 mins followed by substrate addition and measured after 1 hr by chromogeni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635634BDBM50635634(CHEMBL5556274)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-Suc-Ala-Ala-Pro-Phe-pNA as chromogenic substrate incubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635642BDBM50635642(CHEMBL5517985)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-Suc-Ala-Ala-Pro-Phe-pNA as chromogenic substrate incubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635637BDBM50635637(CHEMBL5557890)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-Suc-Ala-Ala-Pro-Phe-pNA as chromogenic substrate incubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120437BDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of chymotrypsin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120426BDBM50120426(CHEMBL3617968)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of chymotrypsin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621710BDBM50621710(CHEMBL5415411)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618526BDBM50618526(CHEMBL5426970)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618526BDBM50618526(CHEMBL5426970)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618540BDBM50618540(CHEMBL5405557)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618528BDBM50618528(CHEMBL5433524)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618530BDBM50618530(CHEMBL5405589)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618554BDBM50618554(CHEMBL5396481)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618548BDBM50618548(CHEMBL5413385)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618551BDBM50618551(CHEMBL5414071)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533256BDBM50533256(CHEMBL4448473)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533253BDBM50533253(CHEMBL4441232)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533253BDBM50533253(CHEMBL4441232)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533254BDBM50533254(CHEMBL4550207)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533254BDBM50533254(CHEMBL4550207)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533256BDBM50533256(CHEMBL4448473)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623332BDBM50623332(CHEMBL5423593)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of chymotrypsin (unknown origin) using N-succinyl-AAPF-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617978BDBM50617978(CHEMBL1488059)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-succinyl-AAPF-AMC as fluorogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617985BDBM50617985(CHEMBL5406478)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Chymotrypsin (unknown origin) using N-succinyl-AAPF-AMC as fluorogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60981BDBM60981(SCH-202676 hydrobromide | SMR001230740 | MLS002153...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of chymotrypsin (unknown origin) using N-succinyl-AAPF-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 513874BDBM513874(bioRxiv20220126.477782, Screening Hit 2 | bioRxiv2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human pancreas chymotrypsin using Suc-Ala-Ala-Pro-Phe-AMC as substrate preincubated for 15 mins incubated followed by addition of subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetChymotrypsinogen B2(Human)
The University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50541448BDBM50541448(CHEMBL4633785)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mammalian chymotrypsin (unknown origin) using Suc-AAPF-AMC as substrate preincubated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed