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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • 5'-AMP-activated protein kinase subunit beta-1
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • CaM kinase I alpha
  • CaM kinase IV
  • Casein kinase I
  • Casein kinase I isoform alpha
  • Casein kinase I isoform delta
  • Casein kinase II subunit alpha
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 6
  • Cyclin-dependent kinase 7
  • Cyclin-dependent kinase 9
  • Cyclin-dependent-like kinase 5
  • Death-associated protein kinase 3
  • Dual specificity protein kinase CLK2
  • Dual specificity protein kinase CLK4
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Dual-specificity tyrosine-phosphorylation regulated kinase 3
  • Ephrin type-A receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 3
  • Glycogen synthase kinase-3
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Inhibitor of nuclear factor kappa-B kinase subunit alpha
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 3
  • MAP kinase-activated protein kinase 5
  • MAP kinase-interacting serine/threonine-protein kinase 2
  • MAP/microtubule affinity-regulating kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Misshapen-like kinase 1
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 13 (MAPK13)
  • Mitogen-activated protein kinase kinase kinase 9 (MLK1)
  • Mitogen-activated protein kinase kinase kinase kinase 2
  • Mixed lineage kinase 7
  • Muscle, skeletal receptor tyrosine protein kinase
  • NUAK family SNF1-like kinase 1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PDZ-binding kinase
  • Protein kinase C (PKC)
  • Protein kinase C delta type
  • Protein kinase C, gamma
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase Src
  • RAC-alpha serine/threonine-protein kinase
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha 4
  • Ribosomal protein S6 kinase alpha 5
  • Ribosomal protein S6 kinase alpha-3
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 31
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase D3
  • Serine/threonine-protein kinase DCLK2
  • Serine/threonine-protein kinase MRCK alpha
  • Serine/threonine-protein kinase Nek11
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase Nek3
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PRKX
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase SRPK3
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase WNK2
  • Serine/threonine-protein kinase c-TAK1
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Testis-specific serine/threonine-protein kinase 1
  • Testis-specific serine/threonine-protein kinase 2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
109 Ki 1 IC50
  • 7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,16-dioxa-2,4,19,21-tetraaza-tricyclo[15.3.1.0*5,10*]henicosa-1(21),5,7,9,17,19-hexaene-18-crbonitrile
  • CHEMBL248757