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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • 1,3-beta-glucan synthase component GLS2
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-1
  • ABL
  • ABL Mutant (E255K)
  • ABL Mutant (F359V)
  • ABL Mutant (H396P)
  • ABL Mutant (M351T)
  • ABL Mutant (Q252H)
  • ABL Mutant (T315I)
  • ABL Mutant (T315N)
  • ABL Mutant (Y253F)
  • ABL1(Q252H)
  • ALK tyrosine kinase receptor
  • AMPK subunit alpha-2
  • AP2-associated protein kinase 1
  • Acetylcholinesterase
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-2A
  • Activin receptor type-2B
  • Activin receptor-like kinase 3 (ALK-3)
  • Angiopoietin-1 receptor
  • Ankyrin repeat and protein kinase domain-containing protein 1
  • Apoptosis Signal-regulating Kinase 1 (ASK1)
  • Aurora Kinase C (Aurora-C)
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • BIKE
  • BMP-2-inducible protein kinase
  • BR serine/threonine-protein kinase 1
  • BR serine/threonine-protein kinase 2
  • BRSK2
  • Bcr-Abl
  • Bile salt export pump
  • Bone Morphogenetic Protein Receptor type II (BMPR2)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Bone morphogenetic protein receptor type-2
  • Bromodomain-containing protein 7
  • Bromodomain-containing protein 9
  • CAMK1D
  • CAMK2A
  • CAMK2B
  • CAMK2G
  • CDC2-like kinase 3 (CLK3)
  • CDKL2
  • CLK1
  • CSNK1A1L
  • CaM kinase I alpha
  • CaM kinase I delta
  • CaM kinase I gamma
  • CaM kinase II
  • CaM kinase IV
  • CaM-kinase kinase alpha
  • CaM-kinase kinase beta
  • Calcium channel (Type L)
  • Calcium-dependent protein kinase 1
  • Calcium/calmodulin-dependent protein kinase type II subunit delta
  • Canalicular multispecific organic anion transporter 1
  • Canalicular multispecific organic anion transporter 2
  • Casein kinase I
  • Casein kinase I isoform alpha
  • Casein kinase I isoform alpha-like
  • Casein kinase I isoform delta
  • Casein kinase I isoform epsilon
  • Casein kinase I isoform gamma-3
  • Casein kinase II subunit alpha
  • Casein kinase II subunit alpha'
  • Cell division control protein 2 homolog
  • Chaperone activity of bc1 complex-like, mitochondrial
  • Citron Rho-interacting kinase
  • Cyclin-dependent kinase 11A
  • Cyclin-dependent kinase 13
  • Cyclin-dependent kinase 15
  • Cyclin-dependent kinase 19
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 3 (CDK3)
  • Cyclin-dependent kinase 4
  • Cyclin-dependent kinase 7
  • Cyclin-dependent kinase 8
  • Cyclin-dependent kinase 9
  • Cyclin-dependent kinase-like 1
  • Cyclin-dependent kinase-like 3
  • Cyclin-dependent kinase-like 5
  • Cyclin-dependent-like kinase 5
  • Cytoplasmic tyrosine-protein kinase BMX
  • DAPK1
  • DCAMKL1
  • DCAMKL2
  • DCAMKL3
  • DLK
  • Death-associated protein kinase 1
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Discoidin domain-containing receptor 2
  • Dual serine/threonine and tyrosine protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 2
  • Dual specificity mitogen-activated protein kinase kinase 3
  • Dual specificity mitogen-activated protein kinase kinase 4
  • Dual specificity mitogen-activated protein kinase kinase 5
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
  • Dual specificity protein kinase CLK1/CLK4
  • Dual specificity protein kinase CLK2
  • Dual specificity protein kinase CLK4
  • Dual specificity protein kinase TTK
  • Dual specificity testis-specific protein kinase 1
  • Dual specificty protein kinase CLK1
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Dual-specificity tyrosine-phosphorylation regulated kinase 2
  • Dual-specificity tyrosine-regulated kinases 1B
  • EBifunctional epoxide hydrolase 2
  • EGF-R Tyrosine Kinase Mutant (G719C)
  • EPHB1
  • Ephrin receptor
  • Ephrin type-A receptor 1 (EPHA1)
  • Ephrin type-A receptor 2
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-A receptor 7
  • Ephrin type-B receptor 2
  • Ephrin type-B receptor 3 (EPHB3)
  • Ephrin type-B receptor 4
  • Epidermal growth factor receptor
  • Epithelial discoidin domain-containing receptor 1
  • Eukaryotic translation initiation factor 2-alpha kinase 1
  • Eukaryotic translation initiation factor 2-alpha kinase 4
  • Extracellular signal-regulated kinase 5 (ERK5)
  • FLT3(D835H)
  • FLT3(D835Y)
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1
  • G protein-coupled receptor kinase 4
  • G protein-coupled receptor kinase 7
  • GCN2(Kin.Dom.2 S808G)
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 1
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Homeodomain-interacting protein kinase 3
  • Homeodomain-interacting protein kinase 4
  • Hormonally up-regulated neu tumor-associated kinase
  • Inhibitor of nuclear factor kappa-B kinase subunit alpha
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin Receptor-Related Protein (INSRR)
  • Insulin receptor
  • Insulin receptor-related protein
  • Insulin-like growth factor I receptor
  • Interferon-induced, double-stranded RNA-activated protein kinase
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 3
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • LIM domain kinase 2
  • Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)
  • Leukocyte tyrosine kinase receptor
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 5
  • MAP kinase-interacting serine/threonine-protein kinase 1
  • MAP kinase-interacting serine/threonine-protein kinase 2
  • MAP/microtubule affinity-regulating kinase 2
  • MAP/microtubule affinity-regulating kinase 4
  • MAP4K1
  • MAP4K5
  • MARK3
  • MARK4
  • MAST1/MAST2
  • MLK1
  • MYO3B
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Macrophage-stimulating protein receptor
  • Mast/stem cell growth factor receptor Kit
  • Maternal embryonic leucine zipper kinase (MELK)
  • Misshapen-like kinase 1
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 11
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 13 (MAPK13)
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 15
  • Mitogen-activated protein kinase 3
  • Mitogen-activated protein kinase 4
  • Mitogen-activated protein kinase 6
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Mitogen-activated protein kinase kinase kinase 1
  • Mitogen-activated protein kinase kinase kinase 10
  • Mitogen-activated protein kinase kinase kinase 11
  • Mitogen-activated protein kinase kinase kinase 12
  • Mitogen-activated protein kinase kinase kinase 13
  • Mitogen-activated protein kinase kinase kinase 15
  • Mitogen-activated protein kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase 4
  • Mitogen-activated protein kinase kinase kinase 6
  • Mitogen-activated protein kinase kinase kinase 7
  • Mitogen-activated protein kinase kinase kinase 9 (MLK1)
  • Mitogen-activated protein kinase kinase kinase kinase 1
  • Mitogen-activated protein kinase kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase kinase 4
  • Mitogen-activated protein kinase kinase kinase kinase 5
  • Mixed lineage kinase 7
  • Multidrug resistance-associated protein 4
  • Muscle, skeletal receptor tyrosine protein kinase
  • Myosin IIIA
  • Myosin light chain kinase
  • Myosin light chain kinase family member 4
  • Myosin light chain kinase, smooth muscle
  • Myosin-IIIB
  • Myotonin-protein kinase
  • NAD-dependent deacetylase sirtuin 2
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • NUAK family SNF1-like kinase 2
  • Non-receptor tyrosine-protein kinase TNK1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PCTK2
  • PCTK3
  • PFTK1
  • PITSLRE serine/threonine-protein kinase CDC2L1
  • PKN1
  • PLK4
  • PRP4 kinase (PRP4)
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
  • Peripheral plasma membrane protein CASK
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • Phosphatidylinositol 4-kinase beta
  • Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta
  • Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma
  • Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha
  • Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma
  • Phosphatidylinositol-5-phosphate 4-kinase type-2 beta
  • Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma
  • Phosphorylase kinase
  • Platelet-derived growth factor receptor alpha
  • Platelet-derived growth factor receptor beta
  • Polo-Like Kinase 3
  • Polo-Like Kinase 4
  • Poly [ADP-ribose] polymerase tankyrase-2
  • Potassium voltage-gated channel subfamily H member 2
  • Protein delta homolog 1
  • Protein kinase C alpha type
  • Protein kinase C delta type
  • Protein kinase C iota (PKCι)
  • Protein kinase C theta type
  • Protein kinase C, epsilon
  • Protein kinase C, eta
  • Protein kinase N1
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase Src
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Putative uncharacterized serine/threonine-protein kinase SgK110
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • RET Mutant (M918T)
  • RPS6KA2(Kin.Dom.2 - C-terminal)
  • RPS6KA4(Kin.Dom.1 - N-terminal)
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Receptor-interacting protein 1 (RIPK1)
  • Receptor-interacting serine/threonine-protein kinase 4
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Rhodopsin kinase
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 4
  • Ribosomal protein S6 kinase alpha 5
  • Ribosomal protein S6 kinase alpha 6
  • Ribosomal protein S6 kinase alpha-3
  • SNF-related serine/threonine-protein kinase
  • SPS1/STE20-related protein kinase YSK4
  • SRPK2
  • STE20/SPS1-related proline-alanine-rich protein kinase
  • Salt-inducible kinase 2 (SIK2)
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 10
  • Serine/threonine-protein kinase 11
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 17B (STK17B)
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase 24
  • Serine/threonine-protein kinase 25
  • Serine/threonine-protein kinase 32A
  • Serine/threonine-protein kinase 32B
  • Serine/threonine-protein kinase 32C
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 35
  • Serine/threonine-protein kinase 36
  • Serine/threonine-protein kinase 38
  • Serine/threonine-protein kinase 38-like
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Aurora-C
  • Serine/threonine-protein kinase B-raf
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D1
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase D3
  • Serine/threonine-protein kinase DCLK1
  • Serine/threonine-protein kinase DCLK2
  • Serine/threonine-protein kinase DCLK3
  • Serine/threonine-protein kinase GAK
  • Serine/threonine-protein kinase ICK
  • Serine/threonine-protein kinase LATS1
  • Serine/threonine-protein kinase LATS2
  • Serine/threonine-protein kinase MAK
  • Serine/threonine-protein kinase MARK1
  • Serine/threonine-protein kinase MRCK alpha
  • Serine/threonine-protein kinase MRCK beta
  • Serine/threonine-protein kinase MRCK gamma
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase NEK7
  • Serine/threonine-protein kinase NEK9
  • Serine/threonine-protein kinase NIM1
  • Serine/threonine-protein kinase Nek1
  • Serine/threonine-protein kinase Nek11
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase Nek3
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase Nek5
  • Serine/threonine-protein kinase OSR1
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PAK7
  • Serine/threonine-protein kinase PCTAIRE-1
  • Serine/threonine-protein kinase PCTAIRE-2
  • Serine/threonine-protein kinase PCTAIRE-3
  • Serine/threonine-protein kinase PFTAIRE-1
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PLK4
  • Serine/threonine-protein kinase PRKX
  • Serine/threonine-protein kinase RIO1
  • Serine/threonine-protein kinase RIO2
  • Serine/threonine-protein kinase RIO3
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase SBK1
  • Serine/threonine-protein kinase SIK1
  • Serine/threonine-protein kinase SIK3
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase SRPK2
  • Serine/threonine-protein kinase SRPK3
  • Serine/threonine-protein kinase Sgk3
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TAO3
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase ULK1
  • Serine/threonine-protein kinase ULK2
  • Serine/threonine-protein kinase ULK3
  • Serine/threonine-protein kinase VRK2
  • Serine/threonine-protein kinase WEE1
  • Serine/threonine-protein kinase c-TAK1
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Serine/threonine-protein kinase pim-3
  • Serine/threonine-protein kinase pknB
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase tousled-like 1
  • Serine/threonine-protein kinase tousled-like 2
  • Serine/threonine-protein kinase/endoribonuclease IRE1 Alpha
  • Sodium channel protein type 5 subunit alpha
  • Solute carrier family 22 member 1
  • TGF-beta receptor type II
  • TLK2
  • TNK1
  • TNNI3K
  • TRAF2 and NCK-interacting protein kinase (TNIK)
  • Testis-specific serine/threonine-protein kinase 1
  • Transient receptor potential cation channel subfamily M member 6
  • Tubulin alpha-1 chain
  • Tyrosine Kinase EPHA3
  • Tyrosine Kinase FLT3 Mutant (N841I)
  • Tyrosine Kinase c-Kit Mutant (N822K)
  • Tyrosine Kinase c-Kit Mutant (V559D)
  • Tyrosine Kinase c-Kit Mutant (V559D/T670I)
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine- and threonine-specific cdc2-inhibitory kinase
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase CTK
  • Tyrosine-protein kinase FER
  • Tyrosine-protein kinase FRK
  • Tyrosine-protein kinase Fes/Fps
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase STK16 (STK16)
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase Srms
  • Tyrosine-protein kinase TEC
  • Tyrosine-protein kinase TXK
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor Tie-1
  • Tyrosine-protein kinase receptor UFO
  • U4/U6 small nuclear ribonucleoprotein Prp4
  • ULK3 kinase
  • Uncharacterized aarF domain-containing protein kinase 4
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • Voltage-gated L-type calcium channel
  • Voltage-gated potassium channel beta subunit Mink/subunit Kv7.1
  • Voltage-gated potassium channel subunit Kv4.3
  • Wee1-like protein kinase 2
  • cAMP-dependent protein kinase (PKA)
  • cGMP-dependent protein kinase
  • cGMP-dependent protein kinase 2
  • myosin light chain kinase 2
  • p21-Activated kinase 2 (PAK2)
  • p21-Activated kinase 3 (PAK3)
38 Ki 158 IC50 1442 Kd 1 EC50
  • CHEMBL535
  • N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
  • N-[2-(diethylamino)ethyl]-5-{[(3Z)-5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-ylidene]methyl}-2,4-dimethyl-1H-pyrrole-3-carboxamide
  • SU11248
  • SUNITINIB
  • SUNITINIB MALATE
  • US10464902, Sunitinib
  • US9163010, Sunitinib
  • US9914707, SU11248