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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-2
  • ALK tyrosine kinase receptor
  • Actin-related protein 2
  • Activin receptor type-1
  • Activin receptor type-1B
  • Aurora kinase A/B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • BR serine/threonine-protein kinase 1
  • BR serine/threonine-protein kinase 2
  • BRAF/CRAF
  • Beta-adrenergic receptor kinase 2
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Bone morphogenetic protein receptor type-2
  • CAMK2A
  • CAMK2B
  • CDC7/Cyclin B1
  • CDK2/CycE
  • CDK2/Cyclin A1
  • CDK3/E
  • CDK4/Cyclin D3
  • CDK6/CycD3
  • CDK7/Cyclin H/MNAT1
  • CDKL2
  • CaM kinase I alpha
  • CaM kinase I delta
  • CaM kinase I gamma
  • CaM kinase II
  • CaM kinase IV
  • CaM-kinase kinase alpha
  • CaM-kinase kinase beta
  • Calcium/calmodulin-dependent protein kinase type 1B
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Casein kinase I
  • Casein kinase I isoform delta
  • Casein kinase I isoform gamma-3
  • Casein kinase II subunit alpha
  • Casein kinase II subunit alpha 3
  • Cereblon/BCR/ABL
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-Y
  • Cyclin-dependent kinase 12
  • Cyclin-dependent kinase 13/Cyclin-K
  • Cyclin-dependent kinase 18
  • Cyclin-dependent kinase-like 1
  • Cyclin-dependent kinase-like 3
  • Cyclin-dependent kinase-like 4
  • Cytoplasmic tyrosine-protein kinase BMX
  • DNA-PK/Ku70/Ku85
  • Death-associated protein kinase 1
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Discoidin domain-containing receptor 2
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
  • Dual specificity mitogen-activated protein kinase kinase; MEK1/2
  • Dual specificity protein kinase CLK1/CLK4
  • Dual specificity protein kinase CLK2
  • Dual specificity protein kinase CLK3
  • Dual specificity protein kinase TTK
  • Dual specificity tyrosine-phosphorylation-regulated kinase 1B
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Dual-specificity tyrosine-phosphorylation regulated kinase 2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 3
  • EPHB1
  • Ephrin receptor
  • Ephrin type-A receptor 2
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-A receptor 7
  • Ephrin type-B receptor 3 (EPHB3)
  • Ephrin type-B receptor 4
  • Epidermal growth factor receptor
  • Eukaryotic elongation factor 2 kinase
  • Eukaryotic translation initiation factor 2-alpha kinase 1
  • Eukaryotic translation initiation factor 2-alpha kinase 4
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
  • G protein-coupled receptor kinase 5
  • G protein-coupled receptor kinase 6
  • G protein-coupled receptor kinase 7
  • G-protein coupled receptor kinase 2
  • Glucokinase/Glucokinase regulatory protein
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 1
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Homeodomain-interacting protein kinase 3
  • Homeodomain-interacting protein kinase 4
  • Inhibitor of NF-kappa-B kinase alpha/beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin receptor-related protein
  • Insulin-like growth factor I receptor
  • Interferon-induced, double-stranded RNA-activated protein kinase
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • LIM domain kinase 2
  • Leucine-rich repeat serine/threonine-protein kinase 2
  • Leukocyte tyrosine kinase receptor
  • MAP kinase-activated protein kinase 3
  • MAP kinase-interacting serine/threonine-protein kinase 1/2
  • MAP/microtubule affinity-regulating kinase 2
  • MAP/microtubule affinity-regulating kinase 3
  • MAP/microtubule affinity-regulating kinase 4
  • MAPK/MAK/MRK overlapping kinase
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Macrophage-stimulating protein receptor
  • Mammalian target of Rapamycin (mTORC1)
  • Mast/stem cell growth factor receptor Kit
  • Maternal embryonic leucine zipper kinase
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 10/Receptor-interacting serine/threonine-protein kinase 1
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase kinase kinase 10
  • Mitogen-activated protein kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase 5
  • Mitogen-activated protein kinase kinase kinase 7
  • Mitogen-activated protein kinase kinase kinase 9
  • Mitogen-activated protein kinase kinase kinase kinase 1
  • Mitogen-activated protein kinase kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase kinase 4
  • Mitogen-activated protein kinase kinase kinase kinase 5
  • Mixed lineage kinase 7
  • Muscle, skeletal receptor tyrosine protein kinase
  • Myosin light chain kinase, smooth muscle
  • Myosin-IIIB
  • Myotonin-protein kinase
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • NUAK family SNF1-like kinase 2
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • PKC alpha and beta-2
  • PRP4 kinase (PRP4)
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
  • Phosphorylase kinase
  • Platelet-derived growth factor receptor
  • Platelet-derived growth factor receptor beta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase C, PKC; classical/novel
  • Protein kinase N1
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Pyruvate dehydrogenase kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • RAF serine/threonine protein kinase
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Rhodopsin kinase
  • Ribosomal protein S6 kinase
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 4
  • Ribosomal protein S6 kinase alpha 6
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine-protein kinase ATM
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 10
  • Serine/threonine-protein kinase 11
  • Serine/threonine-protein kinase 16
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 17B (STK17B)
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase 24
  • Serine/threonine-protein kinase 25
  • Serine/threonine-protein kinase 32A
  • Serine/threonine-protein kinase 32B
  • Serine/threonine-protein kinase 32C
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 35
  • Serine/threonine-protein kinase 38-like
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Aurora-C
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase DCLK2
  • Serine/threonine-protein kinase DCLK3
  • Serine/threonine-protein kinase ICK
  • Serine/threonine-protein kinase MAK
  • Serine/threonine-protein kinase MRCK beta
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase NEK7
  • Serine/threonine-protein kinase NEK9
  • Serine/threonine-protein kinase NIM1
  • Serine/threonine-protein kinase Nek1
  • Serine/threonine-protein kinase Nek11
  • Serine/threonine-protein kinase Nek3
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PAK7
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PRKX
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase SBK1
  • Serine/threonine-protein kinase SIK1
  • Serine/threonine-protein kinase SIK2
  • Serine/threonine-protein kinase SIK3
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase SRPK2
  • Serine/threonine-protein kinase SRPK3
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase Sgk2
  • Serine/threonine-protein kinase Sgk3
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TAO3
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase ULK1
  • Serine/threonine-protein kinase ULK2
  • Serine/threonine-protein kinase ULK3
  • Serine/threonine-protein kinase VRK1
  • Serine/threonine-protein kinase VRK2
  • Serine/threonine-protein kinase WEE1
  • Serine/threonine-protein kinase WNK1
  • Serine/threonine-protein kinase WNK2
  • Serine/threonine-protein kinase WNK3
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Serine/threonine-protein kinase pim-3
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase tousled-like 1
  • Serine/threonine-protein kinase tousled-like 2
  • Serine/threonine-protein kinase/endoribonuclease IRE1 Alpha
  • TGF-beta receptor type II
  • TGF-beta receptor type-1
  • TRAF2- and NCK-interacting kinase
  • Tau-tubulin kinase 1
  • Tau-tubulin kinase 2
  • Testis-specific serine/threonine-protein kinase 1
  • Testis-specific serine/threonine-protein kinase 2
  • Testis-specific serine/threonine-protein kinase 3
  • Testis-specific serine/threonine-protein kinase 4
  • Transcription initiation factor TFIID subunit 1-like
  • Transient receptor potential cation channel subfamily M member 7
  • Tribbles homolog 2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase FER
  • Tyrosine-protein kinase FES
  • Tyrosine-protein kinase FRK
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase TXK
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • Wee1-like protein kinase 2
  • cAMP-dependent protein kinase (PKA)
  • cGMP-dependent protein kinase 1 beta
  • cGMP-dependent protein kinase 2
  • mTOR/FKBP12A/FKBP12B
  • myosin light chain kinase 2
  • p110α/p85α
  • p110β/p85α
  • p21-Activated kinase 3 (PAK3)
  • p38 MAP kinase alpha/beta
  • p38 delta/gamma
361 IC50
  • CHEMBL4438748