Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 1,3-beta-glucan synthase component GLS2
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1A (5HT1A)
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- 5-hydroxytryptamine receptor 7 (5HT7)
- ADRA1A
- ADRA1B
- Adrenergic receptor alpha-1
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- CCKBR
- Calcium channel
- Calcium channel (Type L)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cholecystokinin B
- Cholinergic, muscarinic
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- DRD2
- Delta-type opioid receptor
- Dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Glycine receptor subunit alpha-1
- HTR1D
- HTR2C
- HTR6
- HTR7
- Histamine H1 receptor
- Histone H1
- Kappa-type opioid receptor
- Melanin-concentrating hormone receptor 2/HERG
- Mu-type opioid receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M1 and M3
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- NT
- Norepinephrine Monoamine transporters
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily H member 2
- Prostanoid TP receptor
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sigma non-opioid intracellular receptor 1
- Sodium channel protein type 5 subunit alpha
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
- Solute carrier family 22 member 2
- Substance P
- Transporter
- Voltage-dependent L-type calcium channel subunit alpha-1C
- Voltage-gated L-type calcium channel
- Voltage-gated sodium channel subunit alpha Nav1.8
- adrenergic Alpha2
- (risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
- 1-(2-Allyl-phenoxy)-3-isopropylamino-propan-2-ol
- 2-(2-(4-(benzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-7,8,9,9a-tetrahydro-1H-pyrido[1,2-a]pyrimidin-4(6H)-one
- 2-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-6,7,8,8a-tetrahydro-5H-naphthalen-1-one
- 3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one (Resperidone)
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one (risperidone)
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one(risperidone)
- 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-methyl-1,3-dihydro-indol-2-one(Norastemizole)
- CHEMBL85
- R 64 766
- RISPERDAL
- RISPERIDONE
- US10167256, Risperidone
- US10174011, risperidone
- US10259786, Risperidone
- US10501452, Compound risperidone
- US8802672, Risperidone
- ALK tyrosine kinase receptor
- Angiopoietin-1 receptor
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- BDNF/NT-3 growth factors receptor
- CAMK2B
- Casein kinase I isoform gamma-3
- Cyclin-dependent kinase 1
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 4
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Cytoplasmic tyrosine-protein kinase BMX
- EPHB1
- Ephrin receptor
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Focal adhesion kinase 1
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 5
- MAP kinase-interacting serine/threonine-protein kinase 1
- MAP kinase-interacting serine/threonine-protein kinase 2
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 12
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase 8
- Non-receptor tyrosine-protein kinase TYK2
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Phosphatidylinositol 3-kinase catalytic subunit type 3
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
- Phosphatidylinositol 4-kinase beta
- Platelet-derived growth factor receptor alpha
- Protein kinase C alpha type
- Protein kinase C theta type
- Protein kinase N1
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Receptor tyrosine-protein kinase erbB-2
- Rho-associated protein kinase 2
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase WNK1
- Serine/threonine-protein kinase pim-2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase HCK
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase Mer
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase Yes
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor UFO
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
- p21-Activated kinase 2 (PAK2)
116 IC50
- CHEMBL1834657
- US9434697, BGJ398
- US9730931, BGJ398