Compile Data Set for Download or QSAR
Report error Found 8928 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3'
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149360(Acetic acid 4-(1,4-dioxo-4,5-dihydro-[1,2,4]triazo...)
Affinity DataKi:  4.95E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149367(4-Amino-2-(4-amino-phenyl)-2H-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  3.47E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149356(2-(4-Hydroxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
Affinity DataKi:  4.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149355(2-(4-Nitro-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  6.22E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149368(2-(4-Ethoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]qu...)
Affinity DataKi:  3.75E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149362(4-Amino-2-(4-ethoxy-phenyl)-2H-[1,2,4]triazolo[4,3...)
Affinity DataKi:  3.69E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149358(4-amino-6-nitro-2-phenyl-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  5.32E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149361(4,6-Diamino-2-(4-methoxy-phenyl)-2H-[1,2,4]triazol...)
Affinity DataKi:  4.65E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149369(2-(4-Dimethylamino-phenyl)-2H,5H-[1,2,4]triazolo[4...)
Affinity DataKi:  3.36E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149363(4,6-Diamino-2-(4-hydroxy-phenyl)-2H-[1,2,4]triazol...)
Affinity DataKi:  3.57E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149359(6-Amino-2-(4-methoxy-phenyl)-2H,5H-[1,2,4]triazolo...)
Affinity DataKi:  4.08E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149373(2-(4-Amino-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  2.44E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50086143(4-Amino-2-(4-methoxy-phenyl)-2H-[1,2,4]triazolo[4,...)
Affinity DataKi:  4.34E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149370(4-Amino-2-(4-methoxy-phenyl)-6-nitro-2H-[1,2,4]tri...)
Affinity DataKi:  4.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149357(2-(4-methoxyphenyl)-6-nitro-[1,2,4]triazolo[4,3-a]...)
Affinity DataKi:  5.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50149366(4-Amino-2-(4-hydroxy-phenyl)-2H-[1,2,4]triazolo[4,...)
Affinity DataKi:  4.13E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
Affinity DataKi:  4.79E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067074(1-Chloro-3-pyridin-2-yl-isoquinoline | CHEMBL12851...)
Affinity DataKi:  2.60E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067076(N-(3-Pyridin-2-yl-isoquinolin-1-yl)-formamidine | ...)
Affinity DataKi:  2.00E+7nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067077(TCMDC-123745 | 3-Chloro-N-(3-pyridin-2-yl-isoquino...)
Affinity DataKi:  7.80E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067078(1-Methoxy-3-pyridin-2-yl-isoquinoline | CHEMBL3402...)
Affinity DataKi:  5.60E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067085(N-Acetyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-aceta...)
Affinity DataKi:  3.50E+7nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067083(1-Methanesulfonyl-3-pyridin-2-yl-isoquinoline | CH...)
Affinity DataKi:  1.50E+7nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067087(3,4-Dichloro-N-(3-pyridin-2-yl-isoquinolin-1-yl)-b...)
Affinity DataKi:  2.30E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067086(3-Methyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benza...)
Affinity DataKi:  1.30E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067090(N-(2,6-Dimethyl-benzoyl)-2,6-dimethyl-N-(3-pyridin...)
Affinity DataKi:  3.20E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067073(1-Methylsulfanyl-3-pyridin-2-yl-isoquinoline | CHE...)
Affinity DataKi:  3.90E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067091(3-Pyridin-2-yl-isoquinolin-1-ol | CHEMBL128943)
Affinity DataKi:  2.70E+7nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067072(1-Phenyl-3-pyridin-2-yl-isoquinoline | CHEMBL12884...)
Affinity DataKi:  1.20E+7nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067093(1-Ethyl-3-pyridin-2-yl-isoquinoline | CHEMBL129406)
Affinity DataKi:  5.10E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067094(4-Chloro-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benza...)
Affinity DataKi:  2.30E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067076(N-(3-Pyridin-2-yl-isoquinolin-1-yl)-formamidine | ...)
Affinity DataKi:  2.00E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067104(N-(3-Pyridin-2-yl-isoquinolin-1-yl)-acetamide | CH...)
Affinity DataKi:  1.30E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067091(3-Pyridin-2-yl-isoquinolin-1-ol | CHEMBL128943)
Affinity DataKi:  2.70E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067106(N-(2-Pyridin-2-yl-quinazolin-4-yl)-acetamide | CHE...)
Affinity DataKi:  1.10E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067108(N-(2-Pyridin-2-yl-quinazolin-4-yl)-formamidine | C...)
Affinity DataKi:  4.00E+6nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cells at 10e-5 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067109(2-Pyridin-2-yl-quinazolin-4-ol | CHEMBL128427)
Affinity DataKi:  2.20E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067110(2,6-Dimethyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-b...)
Affinity DataKi:  2.60E+6nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067112(2,2,2-Trifluoro-N-(2-pyridin-2-yl-quinazolin-4-yl)...)
Affinity DataKi:  8.60E+7nMAssay Description:Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50067115(N-(3-Pyridin-2-yl-isoquinolin-1-yl)-isobutyramide ...)
Affinity DataKi:  4.80E+7nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cells at 10e-5 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50088459(1-[2-(4,6-Dimethyl-pyrimidin-2-yl)-quinazolin-4-yl...)
Affinity DataKi:  1.26E+6nMAssay Description:Binding affinity by its ability to displace [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50088461(1-(3-Methoxy-phenyl)-3-(2-phenyl-quinazolin-4-yl)-...)
Affinity DataKi:  2.04E+6nMAssay Description:Binding affinity by its ability to displace [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50088464(1-(2-tert-Butyl-quinazolin-4-yl)-3-phenyl-urea | C...)
Affinity DataKi:  7.87E+7nMAssay Description:Binding affinity by its ability to displace [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50088472(1-phenyl-3-(quinazolin-4-yl)urea | 1-Phenyl-3-quin...)
Affinity DataKi:  1.18E+6nMAssay Description:Binding affinity by its ability to displace [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50009698(CHEMBL48278 | N6-cyclopentyl-9-methyladenine | Cyc...)
Affinity DataKi:  1.33E+6nMAssay Description:Binding affinity against adenosine A3 receptor from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50106536(cid_100053 | 2'-AMINO-2'-DEOXYADENOSINE | 2-aminoa...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50090850((2R,3S,4R,5R)-2-Aminomethyl-5-(6-amino-purin-9-yl)...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50158768(tert-butyl 4-(2-(furan-2-yl)-8-isopentyl-8H-pyrazo...)
Affinity DataKi:  2.51E+6nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50158760(2-Furan-2-yl-8-octyl-8H-pyrazolo[4,3-e][1,2,4]tria...)
Affinity DataKi:  2.04E+6nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50094693(8-tert-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  1.15E+6nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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