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Report error Found 137 Enz. Inhib. hit(s) with Target = 'Galanin receptor type 1'
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50: 0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2018
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307256(Gal(1-13)-Std I | CHEMBL604373 | GWTLNSAGYLLGPrPKP...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | NSC_3043476 | Galantide (M15))
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85200(Galanin rat | Galanin (1-19), rat)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307255(GWTLNSAGYLLGPRHYINLITRQRY-CONH2 | CHEMBL592413)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin rat | Galanin (1-19), rat)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273353((S)-1-(2-((S)-2-((S)-2-((S)-2-(2-((S)-2-((S)-2-((S...)
Affinity DataKi:  0.400nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273366(GWTLNSAGYLLGPHAVGNHRSFSDKNGLT | CHEMBL499179)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293023((Sar)WTLNSAGYLLGPKKKK | CHEMBL508036)
Affinity DataKi:  0.400nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin [D-Trp2], porcine | Galanin (1-29), porcin...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273351(GWTLNSAGYLLGPHAV-NH2 | CHEMBL508083)
Affinity DataKi:  0.5nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293024((Sar)WTLNSAGYLLGPKK(Lys-MPEG4)K | CHEMBL505299)
Affinity DataKi:  0.5nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | NSC_3043476 | Galantide (M15))
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293030((Sar)WTLNSAGYLLGPKK(Lys-octanoyl)K | CHEMBL503900)
Affinity DataKi:  0.700nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273359(CHEMBL526500)
Affinity DataKi:  0.900nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85164(Galanin (1-29), rat)
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | NSC_3043476 | Galantide (M15))
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293029((Sar)WTLNSAGYLLGPKK(Lys-decanoyl)K | CHEMBL460706)
Affinity DataKi:  1.30nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293028((Sar)WTLNSAGYLLGPKK(Lys-lauroyl)K | CHEMBL507733)
Affinity DataKi:  1.40nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307258([N-Ac,des-Sar]Gal-B2 | CHEMBL578317)
Affinity DataKi:  1.70nMAssay Description:Displacement of Eu-labeled galanin from human GalR1 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273354(CHEMBL525755)
Affinity DataKi:  1.90nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50293027((Sar)WTLNSAGYLLGPKK(Lys-myristoyl)K | CHEMBL524678)
Affinity DataKi:  2.60nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273360([Sar1Gly]GAL-B2 | (S)-N-((S)-6-amino-1-((S)-6-amin...)
Affinity DataKi:  2.80nMAssay Description:Displacement of Eu-labeled galanin from human GalR1 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
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