Report error Found 149 Enz. Inhib. hit(s) with Target = 'Low molecular weight protein-tyrosine phosphatase A'
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PtpA assessed as inhibition constant using varying level of pNPP as substrate by Lineweaver-...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv ptpA expressed in Escherichia coli BL21(DE3) using pNPP as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 4.65E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 5.60E+3nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 5.89E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphataseMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA after 20 mins by ELISAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTP-AMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTP-AMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.97E+3nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis H37Rv MptpA using pNPP as substrate incubated for 10 mins and measured by spectrophotometric met...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 9.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.03E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.07E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.14E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-A using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTP-A using p-nitrophenyl phosphate as substrate measured for 10 mins by spectrofluorimetryMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.68E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.79E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.82E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis PtpA using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate a...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.85E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis H37Rv MptpA using pNPP as substrate incubated for 10 mins and measured by spectrophotometric met...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 2.13E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair








































