Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with Target = 'Myeloblastin'
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263166(CHEMBL4071346)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataKi:  6.10nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataKi:  7nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502659(CHEMBL4528256)
Affinity DataKi:  9.80nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataKi:  17nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263172(CHEMBL4085013)
Affinity DataKi:  21nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502657(CHEMBL4589744)
Affinity DataKi:  23nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502654(CHEMBL4470455)
Affinity DataKi:  51nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50270040((S)-1-((1R,2R)-1-cyano-2-phenylcyclopropylamino)-1...)
Affinity DataIC50: 140nMAssay Description:Inhibition of proteinase-3 activation in beta-estradiol differentiated mouse EcoM-G cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMyeloblastin(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50270031(1-((1R,2R)-1-cyano-2-phenylcyclopropylamino)-3-(3-...)
Affinity DataIC50: 150nMAssay Description:Inhibition of proteinase-3 activation in beta-estradiol differentiated mouse EcoM-G cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063047(CHEMBL3398148)
Affinity DataIC50: 220nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50502660(CHEMBL4469546)
Affinity DataKi:  245nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063053(CHEMBL3398164)
Affinity DataIC50: 310nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50084637(Sivelestat | 2,2-Dimethyl-propionic acid 4-[2-(car...)
Affinity DataIC50: 340nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063050(CHEMBL3398145)
Affinity DataIC50: 360nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063052(CHEMBL3398143)
Affinity DataIC50: 470nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50: 530nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101988(CHEMBL3398153)
Affinity DataIC50: 530nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM166437(US9073833, 5)
Affinity DataIC50: 610nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063054(CHEMBL3398165)
Affinity DataIC50: 610nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063051(CHEMBL3398144)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50384111(CHEMBL2029556)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101980(CHEMBL3398150)
Affinity DataIC50: 1.73E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063048(CHEMBL3398147)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101989(CHEMBL3398154)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063049(CHEMBL3398146)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM166438(US9073833, 6)
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50063046(CHEMBL3398149)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101983(CHEMBL3398155)
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263165(CHEMBL4102959)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101984(CHEMBL3398156)
Affinity DataIC50: 3.91E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50269858(Trifluoro-acetate(S)-1-((1S,2S)-1-cyano-2-phenyl-c...)
Affinity DataIC50: 4.55E+3nMAssay Description:Inhibition of proteinase-3 activation in beta-estradiol differentiated mouse EcoM-G cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101978(CHEMBL3398160)
Affinity DataIC50: 4.94E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50384104(CHEMBL2029559)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50444297(CHEMBL3093815)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101981(CHEMBL3398161)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101982(CHEMBL3398162)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50052693((2S,3S)-trans-epoxysuccinyl-L-leucylamido-3-methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of proteinase-3 activation in beta-estradiol differentiated mouse EcoM-G cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101987(CHEMBL3398163)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50266984(CHEMBL4092637)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101985(CHEMBL3398157)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101986(CHEMBL3398158)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PRTN3 (unknown origin) incubated for 1 hr by colloidal coomassie staining based LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50101977(CHEMBL3398159)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50266979(CHEMBL4061897)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50031631(CHEMBL3359767)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetMyeloblastin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM247411(US9453018, 353 | US10336754, Example 353 | US11053...)
Affinity DataKi: >1.20E+4nMAssay Description:Binding affinity to human neutrophil proteinase 3 assessed as inhibition constant using Methoxysuccinyl-L-alanyl-L-alanyl-L-prolylL-valine p-Nitroani...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
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