Affinity DataKi: 0.600nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro inhibition constant for Aurora-CMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:In vitro inhibition constant for Aurora-BMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro inhibition constant for FLT-3More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at integrin alphavbeta3 in human A375M cells assessed as inhibition of cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at integrin alphaVbeta3 in human A375M cells assessed as cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at integrin alphavbeta3 in human A375M cells assessed as inhibition of cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at integrin alpha5beta1 in human A375M cells assessed as inhibition of cell adhesion to fibronectin in presence of Mg2+ and MK-04...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against c-Src kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against c-Src kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against c-Src kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human erbB2 autophosphorylation in MCF7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair