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Found 118 with Last Name = 'lenders' and Initial = 's'
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569962(CHEMBL4864835)
Affinity DataKi:  2.5nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569952(CHEMBL4869028)
Affinity DataKi:  5.5nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569957(CHEMBL4864965)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569960(CHEMBL4852287)
Affinity DataKi:  31nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569963(CHEMBL4855635)
Affinity DataKi:  31nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569958(CHEMBL4864716)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569954(CHEMBL4867227)
Affinity DataKi:  52nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569955(CHEMBL4876966)
Affinity DataKi:  108nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569961(CHEMBL4861722)
Affinity DataKi:  182nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569956(CHEMBL4850408)
Affinity DataKi:  388nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569959(CHEMBL4871282)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544647(CHEMBL4634122)
Affinity DataKi:  2.96E+3nMAssay Description:Inhibition of human neutrophil elastase using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569953(CHEMBL4871079)
Affinity DataKi:  2.97E+3nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544646(CHEMBL4635621)
Affinity DataKi:  2.65E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544646(CHEMBL4635621)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of human neutrophil elastase using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544648(CHEMBL4636971)
Affinity DataKi:  8.38E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584795(CHEMBL5077207)
Affinity DataKd:  2.80E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584796(CHEMBL5094789)
Affinity DataKd:  4.81E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584788(CHEMBL5094633)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584797(CHEMBL5090693)
Affinity DataKd:  3.40E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584798(CHEMBL5075731)
Affinity DataKd:  1.70E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584799(CHEMBL5087113)
Affinity DataKd:  2.04E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584800(CHEMBL5078177)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584801(CHEMBL5091973)
Affinity DataKd:  2.90E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584802(CHEMBL5090725)
Affinity DataKd:  1.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584803(CHEMBL5080701)
Affinity DataKd:  1.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584804(CHEMBL5077431)
Affinity DataKd:  2.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584805(CHEMBL5079115)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584806(CHEMBL5072745)
Affinity DataKd:  1.71E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584807(CHEMBL5076911)
Affinity DataKd:  3.16E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584808(CHEMBL5076160)
Affinity DataKd:  2.46E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584809(CHEMBL5085131)
Affinity DataKd:  2.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584810(CHEMBL5090715)
Affinity DataKd:  2.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584811(CHEMBL5093665)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584812(CHEMBL5072541)
Affinity DataKd:  3.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584813(CHEMBL5089255)
Affinity DataKd:  1.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584814(CHEMBL5081080)
Affinity DataKd:  9.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584815(CHEMBL5086590)
Affinity DataKd:  2.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584816(CHEMBL5087038)
Affinity DataKd:  1.70E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584817(CHEMBL5085870)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584818(CHEMBL5082507)
Affinity DataKd:  3.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584819(CHEMBL5085792)
Affinity DataKd:  1.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584820(CHEMBL5080311)
Affinity DataKd:  2.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584821(CHEMBL5076435)
Affinity DataKd:  3.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584822(CHEMBL5092602)
Affinity DataKd:  41nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584823(CHEMBL5075717)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584824(CHEMBL5080665)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584825(CHEMBL5084413)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584826(CHEMBL5090939)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584827(CHEMBL5082071)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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