Affinity DataKi: 0.0300nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]DAMGO from MOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 168nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 313nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 602nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 793nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.11E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.66E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.82E+5nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.22E+6nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataKd: 8.95E+4nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.00E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+4nMAssay Description:Binding affinity to recombinant rat calcium loaded S100-B by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 4.40E+4nMAssay Description:Binding affinity to recombinant rat calcium loaded S100-B by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 74nMAssay Description:The ability of compounds to protect cells against infection by SARS-CoV-2 is measured by a cell viability assay similar to that described in Weislow,...More data for this Ligand-Target Pair
Affinity DataEC50: 144nMAssay Description:The ability of compounds to protect cells against infection by SARS-CoV-2 is measured by a cell viability assay similar to that described in Weislow,...More data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
Affinity DataKd: 4.60E+3nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.03E+5nMAssay Description:Displacement of TAMRA-TRTK12 from recombinant rat calcium loaded S100-B by Nikolovska-Cleska analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Agonist activity at MOR (unknown origin) by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataEC50: 253nMAssay Description:Agonist activity at MOR (unknown origin) by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair