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Found 34 with Last Name = 'bharti' and Initial = 'sk'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM242374(US10047093, 8-31 | US10392392, Example 8-31 | US10...)
Affinity DataKi:  5nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512177(CHEMBL4451418)
Affinity DataKi:  7.70nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length Pim-1 expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50364776(CHEMBL1952141 | CHEMBL1952329)
Affinity DataKi:  12nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213234(Phen-DC6)
Affinity DataIC50:  0.130nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  0.370nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213233(Telomestatin (TMS))
Affinity DataIC50:  1nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213233(Telomestatin (TMS))
Affinity DataIC50:  1.5nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213233(Telomestatin (TMS))
Affinity DataIC50:  1.90nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213233(Telomestatin (TMS))
Affinity DataIC50:  2nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213233(Telomestatin (TMS))
Affinity DataIC50:  2.20nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  50nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213234(Phen-DC6)
Affinity DataIC50:  55nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512180(CHEMBL4580240)
Affinity DataIC50:  60nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213234(Phen-DC6)
Affinity DataIC50:  60nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  65nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512176(CHEMBL4551767)
Affinity DataIC50:  80nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512179(CHEMBL4469896)
Affinity DataIC50:  111nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213234(Phen-DC6)
Affinity DataIC50:  120nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  130nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512174(CHEMBL4471511)
Affinity DataIC50: <150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512175(CHEMBL4517325)
Affinity DataIC50: <150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM213234(Phen-DC6)
Affinity DataIC50:  174nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  370nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512178(CHEMBL4591510)
Affinity DataIC50:  434nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  1.10E+3nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase DinG(Escherichia coli (Enterobacteria))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  1.20E+3nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  2.30E+3nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)

Curated by ChEMBL
LigandPNGBDBM110190(1-(2,4-Dihydroxyphenyl)-3-(furan-2-yl)propenone (1...)
Affinity DataIC50:  2.49E+3nMAssay Description:Competitive inhibition of PTP1B (unknown origin) using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)

Curated by ChEMBL
LigandPNGBDBM50072958(CHEMBL3410508)
Affinity DataIC50:  2.90E+3nMAssay Description:Competitive inhibition of PTP1B (unknown origin) using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  2.90E+3nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFanconi anemia group J protein(Homo sapiens (Human))
National Institutes of Health, National Institutes of Health Biomedical Research Center

LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  4.90E+3nMpH: 8.0Assay Description:Standard helicase reaction mixtures (20μl) containing 5 fmol of the indicated TP-G4 or OX-1-G2' DNA substrates or forked duplex DNA substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Guru Ghasidas Vishwavidyalaya (A Central University)

Curated by ChEMBL
LigandPNGBDBM50116791(CHEMBL137883)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Guru Ghasidas Vishwavidyalaya (A Central University)

Curated by ChEMBL
LigandPNGBDBM50116790(CHEMBL279386)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)

Curated by ChEMBL
LigandPNGBDBM50121025((E)-1-[2,4-Dihydroxy-5-(3-methyl-but-2-enyl)-pheny...)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed