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Found 147 with Last Name = 'bordeleau' and Initial = 'm'
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  0.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84445(Isoindoline, 12)
Affinity DataKi:  0.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84451(Isoindoline, 18 | Isoindoline, 19)
Affinity DataKi:  0.600nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  1nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84443(Isoindoline, 10 | Isoindoline, 11)
Affinity DataKi:  1.20nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84446(Isoindoline, 13)
Affinity DataKi:  1.20nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84453(Isoindoline, 20)
Affinity DataKi:  1.40nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152303(CHEMBL361035 | N-((S)-1-Benzyl-pyrrolidin-3-yl)-3-...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152303(CHEMBL361035 | N-((S)-1-Benzyl-pyrrolidin-3-yl)-3-...)
Affinity DataKi:  1.5nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152314((S)-N-(1-benzylpyrrolidin-3-yl)-4-(thiophen-2-yl)b...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]ketanserin from cloned human 5HT2A receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152296(CHEMBL364782 | N-((S)-1-Benzyl-pyrrolidin-3-yl)-4-...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152298(CHEMBL426062 | N-((S)-1-Benzyl-pyrrolidin-3-yl)-3-...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152306(CHEMBL187122 | N-(1-Benzyl-pyrrolidin-3-yl)-4-thio...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152297(CHEMBL187236 | N-(1-Benzyl-pyrrolidin-3-yl)-4-thio...)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152314((S)-N-(1-benzylpyrrolidin-3-yl)-4-(thiophen-2-yl)b...)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152314((S)-N-(1-benzylpyrrolidin-3-yl)-4-(thiophen-2-yl)b...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152305(Biphenyl-4-carboxylic acid (1-benzyl-pyrrolidin-3-...)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152302(CHEMBL187113 | N-((R)-1-Benzyl-pyrrolidin-3-yl)-3-...)
Affinity DataKi:  3.40nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84459(Isoindoline, 26)
Affinity DataKi:  3.60nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84449(Isoindoline, 16)
Affinity DataKi:  3.70nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152309(Biphenyl-3-carboxylic acid (1-benzyl-pyrrolidin-3-...)
Affinity DataKi:  4nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174001(CHEMBL381019 | N-[(S)-1-(4-Methyl-benzyl)-pyrrolid...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84456(Isoindoline, 23)
Affinity DataKi:  4.10nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84448(Isoindoline, 15)
Affinity DataKi:  4.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174000((S)-N-(1-(4-fluorobenzyl)pyrrolidin-3-yl)-4-(thiop...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152311(4''-Chloro-biphenyl-4-carboxylic acid (1-benzyl-py...)
Affinity DataKi:  5nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84456(Isoindoline, 23)
Affinity DataKi:  5.30nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174006((S)-N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)pyrrolidi...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152310(4''-Fluoro-biphenyl-4-carboxylic acid (1-benzyl-py...)
Affinity DataKi:  8nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84446(Isoindoline, 13)
Affinity DataKi:  11.9nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84449(Isoindoline, 16)
Affinity DataKi:  12.4nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174000((S)-N-(1-(4-fluorobenzyl)pyrrolidin-3-yl)-4-(thiop...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ketanserin from cloned human 5HT2A receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174003((S)-N-(1-(3-methoxybenzyl)pyrrolidin-3-yl)-4-(thio...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174008((S)-N-(1-(3,4-difluorobenzyl)pyrrolidin-3-yl)-4-(t...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174011((S)-N-(1-(4-(trifluoromethyl)benzyl)pyrrolidin-3-y...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174010((S)-N-(1-(3,4-dichlorobenzyl)pyrrolidin-3-yl)-4-(t...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174008((S)-N-(1-(3,4-difluorobenzyl)pyrrolidin-3-yl)-4-(t...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]ketanserin from cloned human 5HT2A receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174004(CHEMBL197381 | N-((S)-1-(4-chlorobenzyl)pyrrolidin...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152308(4''-Methylsulfanyl-biphenyl-4-carboxylic acid (1-b...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152312(3''-Fluoro-biphenyl-4-carboxylic acid (1-benzyl-py...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152313(4''-Trifluoromethyl-biphenyl-4-carboxylic acid (1-...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84453(Isoindoline, 20)
Affinity DataKi:  17.5nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50152301(CHEMBL366304 | N-((R)-1-Benzyl-pyrrolidin-3-yl)-4-...)
Affinity DataKi:  18nMAssay Description:Ability to displace [3H]-spiperone from human Dopamine receptor D4.2 stably transfected in human embryonic kidney 298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84459(Isoindoline, 26)
Affinity DataKi:  19nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84450(Isoindoline, 17)
Affinity DataKi:  19.1nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84451(Isoindoline, 18 | Isoindoline, 19)
Affinity DataKi:  20nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174002(CHEMBL370652 | N-((S)-1-(4-(trifluoromethyl)benzyl...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174003((S)-N-(1-(3-methoxybenzyl)pyrrolidin-3-yl)-4-(thio...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ketanserin from cloned human 5HT2A receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM50174012((S)-N-(1-(3-(trifluoromethyl)benzyl)pyrrolidin-3-y...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]spiperone from cloned human dopamine D4.2 receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174010((S)-N-(1-(3,4-dichlorobenzyl)pyrrolidin-3-yl)-4-(t...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ketanserin from cloned human 5HT2A receptor in HEK298 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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