TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0450nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 176nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
Affinity DataKi: 183nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 287nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 375nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Neuroscienze Pharmaness S.C.A R.L.
Curated by ChEMBL
Affinity DataKi: 412nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in CD1 mouse brain membrane without cerebellum by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 950nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 2.45E+3nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.83E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 4.25E+3nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in mouse brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in CD1 mouse spleen membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 3.60E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 4.80E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 9.60E+4nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Sassari
Curated by ChEMBL
University Of Sassari
Curated by ChEMBL
Affinity DataKi: 1.10E+5nMAssay Description:Displacement of [125I]alpha-Bungarotoxin from alpha7 nAChR in Sprague-Dawley rat hippocampal membranes pre-incubated for 5 mins followed by overnight...More data for this Ligand-Target Pair