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Found 269 with Last Name = 'cox' and Initial = 'rj'
TargetDihydroxyacetone phosphate acyltransferase(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50068943((S)-2-(3-Carboxy-propionylamino)-6-hydrazino-hepta...)
Affinity DataKi:  22nMAssay Description:Compound was tested for 50% inhibition of N-Succinyl Diaminopimelic Acid Aminotransferase (DAP-AT) from E. coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroxyacetone phosphate acyltransferase(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50068942((S)-2-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataKi:  169nMAssay Description:Compound was tested for binding affinity against N-Succinyl Diaminopimelic Acid Aminotransferase from E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroxyacetone phosphate acyltransferase(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50068940((S)-2-((S)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataKi:  556nMAssay Description:Compound was tested for binding affinity against N-Succinyl Diaminopimelic Acid Aminotransferase from E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Pharmaron-Beijing

Curated by ChEMBL
LigandPNGBDBM50274638(CHEMBL4126156 | US10858355, Example 4)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM50320127(CHEMBL1085565 | N-(3-(1-(2-(4-((N-benzyl-4-chlorop...)
Affinity DataKi:  6.50E+3nMAssay Description:Antagonist activity at CXCR3 (unknown origin) assessed as reduction in CXCL10 induced calcium flux by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target1-deoxy-D-xylulose 5-phosphate reductoisomerase(Escherichia coli)
University of Bristol

LigandPNGBDBM84559(Phosphate analogue, (s)-14)
Affinity DataKi:  7.50E+5nM ΔG°:  -18.6kJ/molepH: 8.0 T: 2°CAssay Description:The assay was monitored spectrophotometrically through the consumption of beta-NADPH. The inhibitor assays contained inhibitor at concentrations of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose 5-phosphate reductoisomerase(Escherichia coli)
University of Bristol

LigandPNGBDBM50032981((3-Amino-propyl)-phosphonic acid | CHEMBL286077 | ...)
Affinity DataKi:  4.00E+6nM ΔG°:  -14.2kJ/molepH: 8.0 T: 2°CAssay Description:The assay was monitored spectrophotometrically through the consumption of beta-NADPH. The inhibitor assays contained inhibitor at concentrations of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose 5-phosphate reductoisomerase(Escherichia coli)
University of Bristol

LigandPNGBDBM84560(Phosphate analogue, (S)-21)
Affinity DataKi:  4.10E+6nM ΔG°:  -14.2kJ/molepH: 8.0 T: 2°CAssay Description:The assay was monitored spectrophotometrically through the consumption of beta-NADPH. The inhibitor assays contained inhibitor at concentrations of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose 5-phosphate reductoisomerase(Escherichia coli)
University of Bristol

LigandPNGBDBM84558(Phosphate analogue, 9)
Affinity DataKi:  6.50E+6nM ΔG°:  -13.0kJ/molepH: 8.0 T: 2°CAssay Description:The assay was monitored spectrophotometrically through the consumption of beta-NADPH. The inhibitor assays contained inhibitor at concentrations of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1-deoxy-D-xylulose 5-phosphate reductoisomerase(Escherichia coli)
University of Bristol

LigandPNGBDBM84557(Phosphate analogue, 6)
Affinity DataKi:  1.80E+7nM ΔG°:  -10.4kJ/molepH: 8.0 T: 2°CAssay Description:The assay was monitored spectrophotometrically through the consumption of beta-NADPH. The inhibitor assays contained inhibitor at concentrations of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50415001(CHEMBL570015 | GSK-256066 | GSK-256066 (3))
Affinity DataIC50: >0.0100nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017300(CHEMBL3287987)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017296(CHEMBL3287739)
Affinity DataIC50:  0.0158nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017308(CHEMBL3287995)
Affinity DataIC50:  0.0158nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017304(CHEMBL3287991)
Affinity DataIC50:  0.0158nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017313(CHEMBL3287999)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human PDE4D using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017307(CHEMBL3287994)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017294(CHEMBL3288029)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human PDE4D using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017335(CHEMBL3288024)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017294(CHEMBL3288029)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of rat PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017338(CHEMBL3288027)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017303(CHEMBL3287990)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017314(CHEMBL3288000)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017298(CHEMBL3288010)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017324(CHEMBL3288012)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017294(CHEMBL3288029)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017301(CHEMBL3287988)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of rat PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017302(CHEMBL3287989)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017311(CHEMBL3287997)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017315(CHEMBL3288001)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017327(CHEMBL3288016)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017333(CHEMBL3288022)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017336(CHEMBL3288025)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017306(CHEMBL3287993)
Affinity DataIC50:  0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017297(CHEMBL3288009)
Affinity DataIC50:  0.0398nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017339(CHEMBL3288028)
Affinity DataIC50:  0.0398nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017319(CHEMBL3288005)
Affinity DataIC50:  0.0501nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017310(CHEMBL3287996)
Affinity DataIC50:  0.0501nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017321(CHEMBL3288006)
Affinity DataIC50:  0.0501nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017312(CHEMBL3287998)
Affinity DataIC50:  0.0501nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017305(CHEMBL3287992)
Affinity DataIC50:  0.0631nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017334(CHEMBL3288023)
Affinity DataIC50:  0.0631nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017299(CHEMBL3288011)
Affinity DataIC50:  0.0631nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017328(CHEMBL3288017)
Affinity DataIC50:  0.0794nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017337(CHEMBL3288026)
Affinity DataIC50:  0.0794nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017326(CHEMBL3288015)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50017331(CHEMBL3288020)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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