Affinity DataKi: 0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]-U69,593 from KOR in guinea pig brain membranes incubated for 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DPDPE from DOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DPDPE from DOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]-U69,593 from KOR in guinea pig brain membranes incubated for 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity to human NPSR by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 59.8nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Displacement of [3H]DPDPE from DOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 169nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Non-competitive inhibition of human PTP1B using p-nitrophenyl phosphate as substrate up to 7 uM preincubated for 10 mins followed by substrate additi...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpB using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: 236nMAssay Description:Displacement of [3H]-U69,593 from KOR in guinea pig brain membranes incubated for 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpB using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
Affinity DataKi: 973nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair