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Found 78 with Last Name = 'gee' and Initial = 'ad'
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249567(CHEMBL4075936)
Affinity DataKi:  25nMAssay Description:Inhibition of CML binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249567(CHEMBL4075936)
Affinity DataKi:  148nMAssay Description:Inhibition of HMGB1 binding to human RAGE domain V expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249567(CHEMBL4075936)
Affinity DataKi:  230nMAssay Description:Inhibition of S110B binding to human RAGE domain V expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataKi:  1.68E+3nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]AVP from human liver vasopressin V1a receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human kidney vasopressin V2 receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249569(CHEMBL4063487)
Affinity DataIC50: <500nMAssay Description:Inhibition of amyloid beta binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249568(CHEMBL4068269)
Affinity DataIC50: <500nMAssay Description:Displacement of [I125]amyloid beta (1 to 40) from human RAGE domain V expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249569(CHEMBL4063487)
Affinity DataIC50: <500nMAssay Description:Inhibition of S110B binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249569(CHEMBL4063487)
Affinity DataIC50: <500nMAssay Description:Inhibition of CML binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249568(CHEMBL4068269)
Affinity DataIC50: <500nMAssay Description:Inhibition of CML binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249568(CHEMBL4068269)
Affinity DataIC50: <500nMAssay Description:Inhibition of S110B binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataIC50:  1.72E+3nMAssay Description:Antagonist activity at human mammary gland oxytocin receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249578(CHEMBL4095634)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of S110B binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50005634(CHEMBL3235375)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of amyloid beta binding to biotin-labeled human RAGE domain V after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249578(CHEMBL4095634)
Affinity DataIC50:  2.29E+3nMAssay Description:Inhibition of amyloid beta binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249578(CHEMBL4095634)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of amyloid beta binding to RAGE (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataIC50:  4.40E+3nMAssay Description:Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataIC50:  7.86E+3nMAssay Description:Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50397836(CHEMBL2179073)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of amyloid beta binding to biotin-labeled human RAGE domain V after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249574(CHEMBL4077165 | US10729695, Compound CB-5)
Affinity DataKd:  1nMAssay Description:Binding affinity to human RAGE cytoplasmic domain by tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249575(CHEMBL4100986 | US10729695, Compound CB-10)
Affinity DataKd:  3nMAssay Description:Binding affinity to human RAGE cytoplasmic domain by tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249576(CHEMBL4075539 | US10729695, Compound CD-6)
Affinity DataKd:  4nMAssay Description:Binding affinity to human RAGE cytoplasmic domain by tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249577(CHEMBL4072531 | US10729695, Compound CB-4)
Affinity DataKd:  2nMAssay Description:Binding affinity to human RAGE cytoplasmic domain by tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249579(CHEMBL1477694 | US10729695, Compound CB-3)
Affinity DataKd:  1nMAssay Description:Binding affinity to human RAGE cytoplasmic domain by tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249580(Azeliragon | PF-04494700 | TTP448 | US11524942, Co...)
Affinity DataKd:  500nMAssay Description:Inhibition of amyloid beta (1 to 42) binding to RAGE domain V (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdvanced glycosylation end product-specific receptor(Homo sapiens (Human))
King'S College London

Curated by ChEMBL
LigandPNGBDBM50249581(CHEBI:6700 | Matrine)
Affinity DataKd:  2.40E+7nMAssay Description:Inhibition of amyloid beta binding to human RAGE domain V (Met1 to Ala 344 residues) expressed in HEK293 cells after 10 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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