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Found 128 with Last Name = 'higaki' and Initial = 'j'
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  4nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  5nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  7nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  10nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  21nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  190nMAssay Description:Inhibition of MMP10More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  660nMAssay Description:Inhibition of MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374977(CHEMBL270849)
Affinity DataIC50:  9nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375063(CHEMBL255607)
Affinity DataIC50:  10nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374956(CHEMBL272978)
Affinity DataIC50:  12nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375073(CHEMBL402340)
Affinity DataIC50:  13nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182409((2R,3S)-N1-((S)-1-(3-(phenylamino)benzyl)-2-oxoaze...)
Affinity DataIC50:  15nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410871(CHEMBL208350)
Affinity DataIC50:  17nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410864(CHEMBL208504)
Affinity DataIC50:  17nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375061(CHEMBL271648)
Affinity DataIC50:  21nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410859(CHEMBL382880)
Affinity DataIC50:  29nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410861(CHEMBL424684)
Affinity DataIC50:  30nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375062(CHEMBL402533)
Affinity DataIC50:  32nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375072(CHEMBL403337)
Affinity DataIC50:  38nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374954(CHEMBL271045)
Affinity DataIC50:  42nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375071(CHEMBL270032)
Affinity DataIC50:  46nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410860(CHEMBL410532)
Affinity DataIC50:  54nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374963(CHEMBL402428)
Affinity DataIC50:  64nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374965(CHEMBL255617)
Affinity DataIC50:  66nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410863(CHEMBL208230)
Affinity DataIC50:  74nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375070(CHEMBL411724)
Affinity DataIC50:  110nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374956(CHEMBL272978)
Affinity DataIC50:  110nMAssay Description:Inhibition of CaMK2delta-mediated vimentin phosphorylation in human HL2 cells after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375077(CHEMBL430412)
Affinity DataIC50:  110nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375064(CHEMBL402152)
Affinity DataIC50:  150nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410868(CHEMBL205970)
Affinity DataIC50:  152nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410867(CHEMBL274414)
Affinity DataIC50:  160nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374966(CHEMBL402524)
Affinity DataIC50:  170nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375069(CHEMBL271426)
Affinity DataIC50:  170nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374989(CHEMBL412302)
Affinity DataIC50:  180nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374989(CHEMBL412302)
Affinity DataIC50:  180nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375067(CHEMBL271043)
Affinity DataIC50:  190nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375080(CHEMBL270141)
Affinity DataIC50:  190nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182403((2R,3S)-N1-((S)-1-(3-phenoxybenzyl)-2-oxoazepan-3-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of beta-amyloid peptide production in CHO N9 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374972(CHEMBL403766)
Affinity DataIC50:  210nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374997(CHEMBL256827)
Affinity DataIC50:  230nMAssay Description:Inhibition of CaMK2delta using 3 weeks old stock solution of compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374952(CHEMBL403054)
Affinity DataIC50:  240nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375066(CHEMBL256460)
Affinity DataIC50:  280nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374988(CHEMBL408434)
Affinity DataIC50:  280nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374960(CHEMBL255633)
Affinity DataIC50:  290nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375001(CHEMBL411253)
Affinity DataIC50:  290nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375054(CHEMBL409856)
Affinity DataIC50:  300nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2695(3-[1-(3-aminopropyl)-1H-indol-3-yl]-4-(1-methyl-1H...)
Affinity DataIC50:  310nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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