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Found 108 with Last Name = 'laneri' and Initial = 's'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM198126((2S,3S,4R,5R)-5-[2-chloro-6-[(3-iodophenyl)methyla...)
Affinity DataKi:  0.220nM ΔG°:  -55.1kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (90 ug) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 5 mM MgCl2, 1 mM EDTA, 2 un...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane after 180 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120763(CHEMBL358076 | Cyclopentanecarboxylic acid (7-ethy...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120761(CHEMBL355898 | Cyclopentanecarboxylic acid (7-meth...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120767(CHEMBL148464 | Cyclopentanecarboxylic acid (7-isop...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120759(CHEMBL146479 | N-(7-Methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  11.8nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120765(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane after 180 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM86761(CAS_35920-39-9 | NECA | NSC_448222)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM86761(CAS_35920-39-9 | NECA | NSC_448222)
Affinity DataKi:  16nM ΔG°:  -44.5kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug) were incubated at 25 °C for 90 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mm MgCl2, 2 units/mL ADA, ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120764(CHEMBL149732 | Cyclopentanecarboxylic acid (2,7-di...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120767(CHEMBL148464 | Cyclopentanecarboxylic acid (7-isop...)
Affinity DataKi:  17.4nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120763(CHEMBL358076 | Cyclopentanecarboxylic acid (7-ethy...)
Affinity DataKi:  20.2nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120766(CHEMBL147582 | N-(2,7-Diphenyl-imidazo[1,2-a][1,3,...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120759(CHEMBL146479 | N-(7-Methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  27.2nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120766(CHEMBL147582 | N-(2,7-Diphenyl-imidazo[1,2-a][1,3,...)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120758(CHEMBL148074 | Cyclopentyl-(7-methyl-2-phenyl-imid...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM86761(CAS_35920-39-9 | NECA | NSC_448222)
Affinity DataKi:  73nM ΔG°:  -40.7kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (90 ug) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 5 mM MgCl2, 1 mM EDTA, 2 un...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  73nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120760(CHEMBL343256 | Cyclohexanecarboxylic acid (7-methy...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493707(CHEMBL2435536)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane after 180 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120760(CHEMBL343256 | Cyclohexanecarboxylic acid (7-methy...)
Affinity DataKi:  202nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120753(CHEMBL421782 | N-(7-Methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  231nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120754(CHEMBL147913 | Cyclohexylmethyl-(7-methyl-2-phenyl...)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  337nM ΔG°:  -36.9kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug) were incubated at 25 °C for 90 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mm MgCl2, 2 units/mL ADA, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493701(CHEMBL2435537)
Affinity DataKi:  343nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane after 180 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  401nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM198126((2S,3S,4R,5R)-5-[2-chloro-6-[(3-iodophenyl)methyla...)
Affinity DataKi:  401nM ΔG°:  -36.5kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug) were incubated at 25 °C for 90 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mm MgCl2, 2 units/mL ADA, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120761(CHEMBL355898 | Cyclopentanecarboxylic acid (7-meth...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120770(Adamantan-1-yl-(7-methyl-2-phenyl-imidazo[1,2-a][1...)
Affinity DataKi:  511nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120770(Adamantan-1-yl-(7-methyl-2-phenyl-imidazo[1,2-a][1...)
Affinity DataKi:  526nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  682nMAssay Description:Displacement of [3H]- CGS-21,680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50120753(CHEMBL421782 | N-(7-Methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  855nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  890nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane after 180 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM198126((2S,3S,4R,5R)-5-[2-chloro-6-[(3-iodophenyl)methyla...)
Affinity DataKi:  890nM ΔG°:  -34.5kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493705(CHEMBL2435534)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493704(CHEMBL2435535)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493703(CHEMBL2435538)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493702(CHEMBL2435540)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493706(CHEMBL2435539)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493707(CHEMBL2435536)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50493701(CHEMBL2435537)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM198129(4-amino-6-alkyloxy-2-benzylthiopyrimidines (6))
Affinity DataKi:  1.20E+3nM ΔG°:  -33.8kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit?? Di Napoli Federico Ii

LigandPNGBDBM50120764(CHEMBL149732 | Cyclopentanecarboxylic acid (2,7-di...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [125I]-AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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