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Found 2195 with Last Name = 'li' and Initial = 'cs'
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557772(CHEMBL4775998)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557773(CHEMBL4778772)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580083(CHEMBL5094268)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580082(CHEMBL5079215)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557775(CHEMBL4758903)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580080(CHEMBL5090624)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580084(CHEMBL5075174)
Affinity DataKi: <0.0500nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557774(CHEMBL4776565)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580081(CHEMBL5094514)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557770(CHEMBL4780060)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557770(CHEMBL4780060)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50096279(CHEMBL3577124)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) using inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50096279(CHEMBL3577124)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557776(CHEMBL4778419)
Affinity DataKi:  0.0620nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580084(CHEMBL5075174)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557770(CHEMBL4780060)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580083(CHEMBL5094268)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580082(CHEMBL5079215)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580081(CHEMBL5094514)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557775(CHEMBL4758903)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557773(CHEMBL4778772)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557772(CHEMBL4775998)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557770(CHEMBL4780060)
Affinity DataKi: <0.0800nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557771(CHEMBL4740241)
Affinity DataKi:  0.0810nMAssay Description:Inhibition of CRAF Y340D/Y341D mutant (unknown origin) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557771(CHEMBL4740241)
Affinity DataKi:  0.102nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557774(CHEMBL4776565)
Affinity DataKi:  0.120nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50096279(CHEMBL3577124)
Affinity DataKi:  0.139nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50096279(CHEMBL3577124)
Affinity DataKi:  0.139nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50580080(CHEMBL5090624)
Affinity DataKi:  0.165nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) inactive MAP2K1 as substrate preincubated for 30 mins measured after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50557776(CHEMBL4778419)
Affinity DataKi:  0.190nMAssay Description:Inhibition of BRAF (unknown origin) (416 to 766) assessed as using inactive phosphorylated MAP2K1 substrate preincubated for 30 mins measured after 9...More data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM349368(US10207991, Ex. Cpd. No. 11 | US10611728, Example ...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM349547(US10207991, Ex. Cpd. No. 62 | US10611728, Example ...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM50577481(CHEMBL4865307)
Affinity DataKi:  9nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM349513(US10207991, Ex. Cpd. No. 28 | US10611728, Example ...)
Affinity DataKi:  11nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataKi:  40nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM50577482(CHEMBL4848550)
Affinity DataKi:  48nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM50577484(CHEMBL4863873)
Affinity DataKi:  50nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM349324(US10207991, Ex. Cpd. No. 8 | US10611728, Example C...)
Affinity DataKi:  79nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Cognition Therapeutics

Curated by ChEMBL
LigandPNGBDBM50577483(CHEMBL4869437)
Affinity DataKi:  120nMAssay Description:Binding affinity to Sigma 2-receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113317(Bis[4-Amino-5-hydroxy-6-(2-methoxy-phenylazo)-naph...)
Affinity DataKi:  190nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50089912((2S)-2-amino-4-methylidenepentanedioic acid | 4-me...)
Affinity DataKi:  3.00E+3nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113314(6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...)
Affinity DataKi:  4.10E+4nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113320(6-(2-Biphenyl-4-yl-vinyl)-quinoline-2,4-dicarboxyl...)
Affinity DataKi:  6.40E+4nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113314(6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...)
Affinity DataKi:  9.50E+4nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113318(6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...)
Affinity DataKi:  1.29E+5nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113321(6-Phenethyl-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  1.43E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113318(6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...)
Affinity DataKi:  1.67E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113323(6-Phenethyloxy-quinoline-2,4-dicarboxylic acid | C...)
Affinity DataKi:  1.89E+5nMAssay Description:Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50113313(4,8-Dihydroxy-quinoline-2-carboxylic acid anion | ...)
Affinity DataKi:  1.90E+5nMAssay Description:Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular glutamate transporter 3(Rattus norvegicus)
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50081123(6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...)
Affinity DataKi:  2.04E+5nMAssay Description:Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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