Compile Data Set for Download or QSAR
maximum 50k data
Found 11 with Last Name = 'mccloud' and Initial = 'tg'
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335578(5'''-episilvestrol | CHEMBL1651030)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335579(17,24-Epoxy-20alpha,25-dihydroxy-21-norbaccharan-3...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335580(20R,24S-Epoxy-25-hydroxy-A-homo-4-oxadammaran-3-on...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335581(20S,24S-Epoxy-25-hydroxy-A-homo-4-oxadammaran-3-on...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335582(4,6-Diene-1beta,15-dihydroxyeudesma-3-one | CHEMBL...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50335583(CHEMBL555196 | silvestrol)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of NFkappaB p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by che...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50480586(CHEMBL553660)
Affinity DataEC50:  600nMAssay Description:Inhibition of HIF1 activation in human U251 cells stably transfected in pGL2-TK-HRE plasmid under hypoxic condition after 16 to 24 hrs by luciferase ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataEC50:  120nMAssay Description:Inhibition of HIF1 activation in human U251 cells stably transfected in pGL2-TK-HRE plasmid under hypoxic condition after 16 to 24 hrs by luciferase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50480587(CHEBI:27663 | Convallatoxin)
Affinity DataEC50:  20nMAssay Description:Inhibition of HIF1 activation in human U251 cells stably transfected in pGL2-TK-HRE plasmid under hypoxic condition after 16 to 24 hrs by luciferase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50480588(CHEMBL538442 | K-Strophanthoside)
Affinity DataEC50:  40nMAssay Description:Inhibition of HIF1 activation in human U251 cells stably transfected in pGL2-TK-HRE plasmid under hypoxic condition after 16 to 24 hrs by luciferase ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50255120(CHEBI:38178 | STROPHANTHIDIN)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of HIF1 activation in human U251 cells stably transfected in pGL2-TK-HRE plasmid under hypoxic condition after 16 to 24 hrs by luciferase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed