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Found 328 with Last Name = 'parrill' and Initial = 'al'
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176394(CHEMBL202361 | octanoic acid (R)-2-octanoyloxy-3-t...)
Affinity DataKi:  5nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271765(3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phen...)
Affinity DataKi:  7.20nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271763(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Affinity DataKi:  20.8nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271764(3-[4'-(3-Carboxy-acryloylamino)-biphenyl-4-ylcarba...)
Affinity DataKi:  21.1nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176391(CHEMBL202185 | octanoic acid (R)-2-octanoyloxy-3-p...)
Affinity DataKi:  39nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)
Affinity DataKi:  48nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271763(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Affinity DataKi:  50nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176397(CHEMBL203986 | nonanoic acid (S)-2-nonanoyloxy-3-p...)
Affinity DataKi:  50nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataKi:  100nMAssay Description:Noncompetitive type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439703(CHEMBL2418930)
Affinity DataKi:  100nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176392(CHEMBL379248 | thiophosphoric acid (R)-2-octanoyla...)
Affinity DataKi:  118nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176393(CHEMBL383095 | octanoic acid (S)-2-octanoyloxy-3-p...)
Affinity DataKi:  119nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176398((S)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosp...)
Affinity DataKi:  139nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176396(CHEMBL204037 | Serine amide phospate derivative | ...)
Affinity DataKi:  196nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300224(4-amino-4-(hydroxymethyl)-6-(4-octylphenyl)hexylph...)
Affinity DataKi:  200nMAssay Description:Noncompetitive type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439704(CHEMBL2418934)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176393(CHEMBL383095 | octanoic acid (S)-2-octanoyloxy-3-p...)
Affinity DataKi:  221nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)
Affinity DataKi:  230nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50316078((5-amino-3-((4'-((8-amino-1-hydroxy-3,6-disulfo-2-...)
Affinity DataKi:  271nMAssay Description:Competitive inhibition of human recombinant C-terminal FLAG-tagged autotaxin expressed in baculovirus-infected Sf9 cells assessed as FS-3 hydrolysis ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 5(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)
Affinity DataKi:  292nMAssay Description:Binding affinity to LPA5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50271765(3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phen...)
Affinity DataKi:  310nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50304581(2-(1,3-dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic ...)
Affinity DataKi:  311nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50241460(4-(3-benzamidophenylamino)-4-oxobut-2-enoic acid |...)
Affinity DataKi:  317nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176394(CHEMBL202361 | octanoic acid (R)-2-octanoyloxy-3-t...)
Affinity DataKi:  360nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176391(CHEMBL202185 | octanoic acid (R)-2-octanoyloxy-3-p...)
Affinity DataKi:  407nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176395(CHEMBL202251 | phosphoric acid mono-((R)-2-octanoy...)
Affinity DataKi:  489nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50176395(CHEMBL202251 | phosphoric acid mono-((R)-2-octanoy...)
Affinity DataKi:  489nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439705(CHEMBL2418932)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300212(2-(4-{[(3-Trifluoromethylphenyl)amino]carbonothioy...)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50332461((R)-3-carba cyclic-phosphatidic acid | CHEMBL16300...)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant ATX mediated hydrolysis of FS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439706(CHEMBL2418933)
Affinity DataKi:  800nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataKi:  824nMAssay Description:Competitive inhibition of human recombinant C-terminal FLAG-tagged autotaxin expressed in baculovirus-infected Sf9 cells assessed as FS-3 hydrolysis ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50304581(2-(1,3-dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic ...)
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50316087(7-[(4-{[4-({4-[(6,8-disulfonaphthalen-2-yl)carbamo...)
Affinity DataKi:  1.14E+3nMAssay Description:Competitive inhibition of human recombinant C-terminal FLAG-tagged autotaxin expressed in baculovirus-infected Sf9 cells assessed as FS-3 hydrolysis ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50316081(5-amino-2-((4'-((6-amino-3-hydroxy-1-sulfonaphthal...)
Affinity DataKi:  1.46E+3nMAssay Description:Competitive inhibition of human recombinant C-terminal FLAG-tagged autotaxin expressed in baculovirus-infected Sf9 cells assessed as FS-3 hydrolysis ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-chimaerin(Homo sapiens (Human))
University Of Tennessee College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50098227(CHEMBL275750 | Pentanoic acid 2-[4-(3-benzylamino-...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity of the compound towards beta chimerinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439709(CHEMBL2418931)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50332460((S)-carba cyclic-phosphatidic acid | CHEMBL1630084)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant ATX mediated hydrolysis of FS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50439708(CHEMBL2418939)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive inhibition of C-terminal FLAG-tagged human recombinant autotaxin using synthetic substrate FS-3 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50079267(Congo Red | Direct red 28 | Kongorot | Sodium diph...)
Affinity DataKi:  1.89E+3nMAssay Description:Noncompetitive inhibition of human recombinant C-terminal FLAG-tagged autotaxin expressed in baculovirus-infected Sf9 cells assessed as FS-3 hydrolys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tennessee College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50098227(CHEMBL275750 | Pentanoic acid 2-[4-(3-benzylamino-...)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity for Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300210(2-(4-{[(3-Chlorophenyl)amino]carbonothioyl}-1-pipe...)
Affinity DataKi:  2.60E+3nMAssay Description:Mixed type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataKi:  2.70E+3nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataKi:  2.70E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tennessee College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50098227(CHEMBL275750 | Pentanoic acid 2-[4-(3-benzylamino-...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity for PKC-delta C1bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176392(CHEMBL379248 | thiophosphoric acid (R)-2-octanoyla...)
Affinity DataKi:  2.85E+3nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50176392(CHEMBL379248 | thiophosphoric acid (R)-2-octanoyla...)
Affinity DataKi:  2.85E+3nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300209(2-(4-{[(2,5-Dichlorophenyl)amino]carbonothioyl}-1-...)
Affinity DataKi:  3.40E+3nMAssay Description:Mixed type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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