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Found 88 with Last Name = 'peeters' and Initial = 't'
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50002694(MOTILIN)
Affinity DataKi:  0.360nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85994([leu13]pMOT(1-19))
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85979([ala3,leu13]pMOT(1-14))
Affinity DataKi:  1.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85987([leu13]pMOT(1-16))
Affinity DataKi:  2.14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  2.82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85981([ala1,leu13]pMOT(1-14) | [leu13]pMOT(1-14))
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85986([ala11,leu13]pMOT(1-14))
Affinity DataKi:  4.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85992([ala10,leu13]pMOT(1-14))
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85989(N-ethyl, N-methyl Erythromycin-A enol ether)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85980([ala12,leu13]pMOT(1-14))
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85999([ala14,leu13]pMOT(1-14))
Affinity DataKi:  7.08nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85990([ala13,leu13]pMOT(1-14))
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85993(Erythromycin-B enol ether)
Affinity DataKi:  7.59nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199368((9R,12R,15S)-12-isopropyl-9-(4-methoxy-benzyl)-15-...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199372((9R,12R,15S)-12-isopropyl-9-naphthalen-1-ylmethyl-...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  8.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199359((9R,12R,15S)-9-benzo[b]thiophen-3-ylmethyl-12-isop...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85984([ala5,leu13]pMOT(1-14))
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85983([ala8,leu13]pMOT(1-14))
Affinity DataKi:  36.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85978([ala6,leu13]pMOT(1-14))
Affinity DataKi:  46.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199397((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199347((9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8...)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86685(ABT-229)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199353((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-i...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85991([ala9,leu13]pMOT(1-14))
Affinity DataKi:  75.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199373((9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199396((9R,12R,15S)-12-isopropyl-9-naphthalen-2-ylmethyl-...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85995([leu13]pMOT(1-11))
Affinity DataKi:  89.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataKi:  137nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85998(Erythromycin-B)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199362((9R,12R,15S)-15-benzyl-9-(4-hydroxy-benzyl)-12-iso...)
Affinity DataKi:  185nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199394((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  192nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199364((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-methyl-15-pro...)
Affinity DataKi:  196nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199392((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-i...)
Affinity DataKi:  222nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85988(N-ethyl, N-Methyl Erythromycin-A)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199346((9R,12R,15S)-9-(1H-indol-3-ylmethyl)-12-isopropyl-...)
Affinity DataKi:  255nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86688(EM-B enolether)
Affinity DataKi:  324nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199390((9R,12R,15R)-9-(4-Hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  335nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86686(Erythromycin A Enol Ether | ME4)
Affinity DataKi:  537nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85981([ala1,leu13]pMOT(1-14) | [leu13]pMOT(1-14))
Affinity DataKi:  589nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199376((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-hydroxymethyl...)
Affinity DataKi:  650nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199378((9R,12R,15S)-15-(4-amino-butyl)-9-(4-hydroxy-benzy...)
Affinity DataKi:  664nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199349((E)-(3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-...)
Affinity DataKi:  701nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199361((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  982nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199360((3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-prop...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199351((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85982([ala7,leu13]pMOT(1-14))
Affinity DataKi:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199363((9R,12R,15S)-12-isopropyl-9-phenethyl-15-propyl-6,...)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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