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Found 61 with Last Name = 'rotondaro' and Initial = 'l'
TargetSubstance-K receptor(Homo sapiens (Human))
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LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473829(CHEMBL389459 | MEN-11995)
Affinity DataKi:  0.158nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473828(CHEMBL116812 | MEN-11990)
Affinity DataKi:  0.316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473824(CHEMBL406024 | MEN-11959)
Affinity DataKi:  0.398nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50366377(CHEMBL334721 | MEN-10627)
Affinity DataKi:  0.631nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473818(CHEMBL406287 | MEN-11842)
Affinity DataKi:  0.794nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473833(CHEMBL420859 | MEN-11830)
Affinity DataKi:  1.60nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472917(CHEMBL323884 | MEN-11749)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472917(CHEMBL323884 | MEN-11749)
Affinity DataKi:  1.60nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50404020(CHEMBL435324 | MEN-11558)
Affinity DataKi:  2nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50404020(CHEMBL435324 | MEN-11558)
Affinity DataKi:  2nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKi:  2.5nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473823(CHEMBL420308 | MEN-11691)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473822(CHEMBL438559 | MEN-11799)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473836(CHEMBL324313 | MEN-11701)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473830(CHEMBL323677 | MEN-11703)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473839(CHEMBL116871 | MEN-11987)
Affinity DataKi:  4nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473821(CHEMBL114068 | MEN-11986)
Affinity DataKi:  4nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473825(CHEMBL113765 | MEN-11983)
Affinity DataKi:  5nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473831(CHEMBL432986 | MEN-11757)
Affinity DataKi:  6.30nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472912(CHEMBL116564 | MEN-11712)
Affinity DataKi:  7.90nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472912(CHEMBL116564 | MEN-11712)
Affinity DataKi:  7.90nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473837(CHEMBL324532 | MEN-11877)
Affinity DataKi:  7.90nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472908(CHEMBL336053)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472910(CHEMBL263194)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473838(CHEMBL116629 | MEN-11708)
Affinity DataKi:  10nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473827(CHEMBL323836 | MEN-11668)
Affinity DataKi:  13nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473832(CHEMBL116969 | MEN-11755)
Affinity DataKi:  13nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472913(CHEMBL2112675)
Affinity DataKi:  20nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473834(CHEMBL324106 | MEN-11733)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473826(CHEMBL116855 | MEN-11715)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472914(CHEMBL114442 | MEN-11667)
Affinity DataKi:  316nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472914(CHEMBL114442 | MEN-11667)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473820(CHEMBL117039 | MEN-11716)
Affinity DataKi:  398nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50473819(CHEMBL326790 | MEN-11532)
Affinity DataKi:  631nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472919(CHEMBL337628)
Affinity DataKi:  631nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472915(CHEMBL114036 | MEN-11540)
Affinity DataKi:  794nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472915(CHEMBL114036 | MEN-11540)
Affinity DataKi:  794nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472918(CHEMBL324804 | MEN-11970)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472907(CHEMBL131024)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472918(CHEMBL324804 | MEN-11970)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472909(CHEMBL2112669)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472906(CHEMBL2111858)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473835(CHEMBL420685 | MEN-11523)
Affinity DataKi:  3.98E+3nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKd:  1.90nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr206Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKd:  26nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50404020(CHEMBL435324 | MEN-11558)
Affinity DataKd:  34nMAssay Description:Compound was evaluated for Kd value against [125I]NKA on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKd:  291nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Phe270Ala mutated human NK-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKd:  48nMAssay Description:Compound was evaluated for Kd value against [3H]-SR- 48968 on the Tyr266Phe mutated human NK-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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