Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 97nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.60E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.60E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.80E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >4.40E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >4.50E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Displacement of [3H]-spiperone from human dopamine receptor subtype hD3 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.360nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 510nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 1.90nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 35nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 4.20nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.820nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.650nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.25nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.660nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 0.150nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit PEN-2/Nicastrin [34-709]/Presenilin-1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 10.7nMAssay Description:A whole-cell gamma-secretase inhibition assay using SHSY5Y neuroblastoma cells in which human gamma-secretase catalyzes the breakdown of the overexpr...More data for this Ligand-Target Pair