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Found 423 with Last Name = 'wilkes' and Initial = 'bc'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008834(CHEMBL3236671)
Affinity DataKi:  0.00935nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  0.0240nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198754(CHEMBL3924888)
Affinity DataKi:  0.0323nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198760(CHEMBL3897031)
Affinity DataKi:  0.0637nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198758(CHEMBL3908315)
Affinity DataKi:  0.0745nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008837(CHEMBL3236674)
Affinity DataKi:  0.0958nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008840(CHEMBL3236677)
Affinity DataKi:  0.0991nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008838(CHEMBL3236675)
Affinity DataKi:  0.109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001157(CHEMBL538700)
Affinity DataKi:  0.118nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198755(CHEMBL3979449)
Affinity DataKi:  0.124nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008841(CHEMBL3236678)
Affinity DataKi:  0.143nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198757(CHEMBL363142)
Affinity DataKi:  0.143nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50493138(CHEMBL3038186)
Affinity DataKi:  0.146nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50493134(CHEMBL3038184)
Affinity DataKi:  0.146nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008836(CHEMBL3236673)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008835(CHEMBL3236672)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.182nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008839(CHEMBL3236676)
Affinity DataKi:  0.235nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008836(CHEMBL3236673)
Affinity DataKi:  0.236nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299557((S)-2-((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50493137(CHEMBL3038180)
Affinity DataKi:  0.306nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  0.308nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM85328(TIPP-PSI | TIPPpsi)
Affinity DataKi:  0.308nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  0.308nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50493132(CHEMBL3038179)
Affinity DataKi:  0.354nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50080453((S)-2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  0.447nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50314880(CHEMBL1089542 | N-(3-(guanidinomethyl)benzyl)-N-(1...)
Affinity DataKi:  0.448nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299558(CHEMBL583488 | H-4'-carboxamido-2',6'-dimethylphen...)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50493134(CHEMBL3038184)
Affinity DataKi:  0.518nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50314880(CHEMBL1089542 | N-(3-(guanidinomethyl)benzyl)-N-(1...)
Affinity DataKi:  0.536nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299559(CHEMBL583285 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.536nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299560(CHEMBL572542 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.605nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL220333 | CHEMBL223244 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  0.616nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299561(CHEMBL572543 | H-4'-[N-((4'-phenyl)phenethyl)carbo...)
Affinity DataKi:  0.646nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001456(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  0.665nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198754(CHEMBL3924888)
Affinity DataKi:  0.733nMAssay Description:Displacement of [3H]U69,593 from KOR in guinea pig brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299562(CHEMBL572494 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  0.783nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198755(CHEMBL3979449)
Affinity DataKi:  0.786nMAssay Description:Displacement of [3H]U69,593 from KOR in guinea pig brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50493133(CHEMBL3038185)
Affinity DataKi:  0.789nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50198754(CHEMBL3924888)
Affinity DataKi:  0.807nMAssay Description:Displacement of [3H]DSLET from DOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataKi:  0.822nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299563(CHEMBL583487 | H-2',6'-dimethyl-4'-[N-((4'-phenyl)...)
Affinity DataKi:  0.825nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50080453((S)-2-({2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKi:  0.943nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50008837(CHEMBL3236674)
Affinity DataKi:  0.961nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig brain membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50493135(CHEMBL3038182)
Affinity DataKi:  0.968nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50007327(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  0.981nMAssay Description:Displacement of [3H]-DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50493133(CHEMBL3038185)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50198752(CHEMBL3976694)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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