Affinity DataKi: 0.190nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]- NECA antagonism of adenylate cyclase activation in human plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of adenylate cyclase via A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against high affinity component of adenosine A1 receptors from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat fat cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity for adenosine A2 receptor using [3H]- NECA antagonism of adenylate cyclase activation in human plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity against low affinity component of adenosine A1 receptors from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 50nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity against low affinity component of Adenosine A1 receptor from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 159nMAssay Description:Binding affinity against high affinity component of Adenosine A1 receptor from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity against A2 adenosine receptor in [3H]adenine-labeled guinea pig cerebral cortical slicesMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to A1 adenosine receptor in rat fat cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity towards Adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity towards Adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity against A2 adenosine receptor in guinea pig cerebral cortical slices by [3H]-adenine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity towards Adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity for adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity for adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranesMore data for this Ligand-Target Pair
