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TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315584(7-Amino-5-dimethylammino-2-(2-furyl)-[1,2,4]triazo...)
Affinity DataEC50:  3.37E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315585(7-Diphenyl-acetylamino-2-(2-furyl)-5-methylthio[1,...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315586(2-(2-Furyl)-5-methylthio-7-phenylacetylamino[1,2,4...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315587(2-(2-Furyl)-7-[4-(methoxyphenyl)acetyl]amino-5-met...)
Affinity DataEC50:  4.24E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315588(2-(2-Furyl)-5-methylthio-7-n-pentylcarbonylamino-[...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315589(1-(2-(furan-2-yl)-5-(methylthio)-[1,2,4]triazolo[1...)
Affinity DataEC50:  1.71E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315590(1-(2-(furan-2-yl)-5-(methylthio)-[1,2,4]triazolo[1...)
Affinity DataEC50:  1.68E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315591(7-Diphenylacetylamino-2-(2-furyl)-5-phenoxy[1,2,4]...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315592(2-(2-Furyl)-5-phenoxy 7-phenylacetylamino-[1,2,4]t...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315593(2-(2-Furyl)-7-[4-(methoxyphenyl)acetyl]amino-5-phe...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315594(2-(2-Furyl)-7-n-pentylcarbonylamino-5-phenoxy[1,2,...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315595(N-(2-(furan-2-yl)-5-phenoxy-[1,2,4]triazolo[1,5-a]...)
Affinity DataEC50:  8.87E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315596(1-(2-(furan-2-yl)-5-phenoxy-[1,2,4]triazolo[1,5-a]...)
Affinity DataEC50:  2.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315597(5-Dimethylamino-7-diphenylacetylamino-2-(2-furyl)-...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315598(5-Dimethylamino-2-(2-furyl)-7-phenylacetylamino-[1...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315599(5-Dimethylamino-2-(2-furyl)-7-[4-(methoxyphenyl)-a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315600(5-Dimethylamino-2-(2-furyl)-7-n-pentylcarbonylamin...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315601(1-(5-(dimethylamino)-2-(furan-2-yl)-[1,2,4]triazol...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315602(1-(5-(dimethylamino)-2-(furan-2-yl)-[1,2,4]triazol...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315603(2-(furan-2-yl)-5-phenoxy-[1,2,4]triazolo[1,5-a][1,...)
Affinity DataEC50:  3.42E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315604(2-(furan-2-yl)-5-(methylthio)-[1,2,4]triazolo[1,5-...)
Affinity DataEC50:  1.49E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50117108(4-[3-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataIC50: 2nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109454(1-(4-Chloro-phenyl)-3-(2-furan-2-yl-8-methyl-8H-py...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptor; range 1.2-4.9More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109434(1-(4-Fluoro-phenyl)-3-(2-furan-2-yl-8-methyl-8H-py...)
Affinity DataIC50: 3nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 2.0-4.3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109441(1-(benzo[d][1,3]dioxol-5-yl)-3-(2-(furan-2-yl)-8-m...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 1.8-5.6More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 2.7-6.6More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109472(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 2.7-7.8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109451(1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109487(1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 3.0-10.8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109453(N-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109468(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 3.7-117More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109474(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 5.5-10.9More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109459(1-(2-chlorophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-p...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 4.4-15.2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109443(1-(3,4-dichlorophenyl)-3-(2-(furan-2-yl)-8-methyl-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 15-44More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133368(N-(2-(furan-2-yl)-8-(3-phenylpropyl)-8H-pyrazolo[4...)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133367(N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133365(N-[2-Furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133361(N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3...)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133360(N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133366(N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50109450(4-(3-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1...)
Affinity DataIC50: 190nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 130-279More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133362(N-[2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133363(N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50183520(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 244nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50133364(N-[2-Furan-2-yl-8-(3-phenyl-propyl)-8H-pyrazolo[4,...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50183529(5-[[(benzofuran-2-yl)amino]carbonyl]amino-8-methyl...)
Affinity DataIC50: 250nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50183527(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 260nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50183526(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 280nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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