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Found 19 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50039218
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317865(2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole |...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321813(4-((1H-Imidazol-4-yl)methyl)-1-(3-isopropylphenyl)...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321823(4-((1H-Imidazol-4-yl)methyl)-1-(3-(trifluoromethyl...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321827(4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N,N...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321826(4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N-m...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321815(4-((1H-Imidazol-4-yl)methyl)-1-(4-(trifluoromethyl...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321816(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321821(4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)pip...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321824(4-((1H-Imidazol-4-yl)methyl)-1-(4-isopropylphenyl)...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321825(4-((1H-Imidazol-4-yl)methyl)-1-(4-tert-butylphenyl...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321828(4-((1H-Imidazol-4-yl)methyl)-1-(naphthalen-2-yl)pi...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321822(4-((1H-Imidazol-4-yl)methyl)-1-(4-nitrophenyl)pipe...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321820(4-((1H-Imidazol-4-yl)methyl)-1-phenylpiperidine | ...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321814(4-((1H-Imidazol-4-yl)methyl)-1-(biphenyl-4-yl)pipe...)
Affinity DataKi:  61nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321829(3-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)pyri...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321817(1-((1H-Imidazol-4-yl)methyl)-4-phenylpiperazine | ...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321819(1-((1H-Imidazol-4-yl)methyl)-4-(4-tert-butylphenyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321818(1-((1H-Imidazol-4-yl)methyl)-4-(4-trifluoromethylp...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed