TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.310nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.490nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.620nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.870nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.880nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 0.890nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 3.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 7.20nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 8.80nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University of California Irvine
Curated by PDSP Ki Database
University of California Irvine
Curated by PDSP Ki Database
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
