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Report error Found 129 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 2'
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50596196(CHEBI:16978 | CHEMBL451509)
Affinity DataEC50:  8.90nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50297387((5S-(5R*,6S*(S*),7E,9E,11Z,14Z))-6-((2-Amino-2-car...)
Affinity DataEC50:  293nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066948(CHEMBL3403187)
Affinity DataIC50: 0.310nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066911(CHEMBL3401689)
Affinity DataIC50: 0.490nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033089(CHEMBL3342959)
Affinity DataIC50: 0.620nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033094(CHEMBL3342964)
Affinity DataIC50: 0.870nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104905(CHEMBL3597618)
Affinity DataIC50: 0.880nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104883(CHEMBL3597616)
Affinity DataIC50: 0.890nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104867(CHEMBL3597530)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104869(CHEMBL3597532)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104839(CHEMBL3597525)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104870(CHEMBL3597533)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033085(CHEMBL3342955)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033085(CHEMBL3342955)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033085(CHEMBL3342955)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066947(CHEMBL3403186)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104918(CHEMBL3597631)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104868(CHEMBL3597531)
Affinity DataIC50: 3.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104864(CHEMBL3597527)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104865(CHEMBL3597528)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104872(CHEMBL3597535)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104911(CHEMBL3597624)
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066942(CHEMBL3401691)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066908(CHEMBL3401687)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104904(CHEMBL3597617)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104836(CHEMBL3597522)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104871(CHEMBL3597534)
Affinity DataIC50: 7.20nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Guinea pig)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50104921(CHEMBL3597634)
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104920(CHEMBL3597633)
Affinity DataIC50: 8.80nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Guinea pig)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50104918(CHEMBL3597631)
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Guinea pig)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50104919(CHEMBL3597632)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104915(CHEMBL3597628)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Guinea pig)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50104920(CHEMBL3597633)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104919(CHEMBL3597632)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104840(CHEMBL3597526)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066946(CHEMBL3403185)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104866(CHEMBL3597529)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104910(CHEMBL3597623)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033091(CHEMBL3342961)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066941(CHEMBL3401690)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066909(CHEMBL3401688)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50033092(CHEMBL3342962)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104908(CHEMBL3597621)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104838(CHEMBL3597524)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Guinea pig)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50104911(CHEMBL3597624)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at guinea pig CysLT2 expressed in CHOK1 cells assessed as inhibition of LTC4-induced calcium mobilization preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50066952(CHEMBL3403190)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104837(CHEMBL3597523)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50104921(CHEMBL3597634)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
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