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Found 289 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 4'
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237577(CHEMBL4087247)
Affinity DataIC50:  233nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237575(CHEMBL4094930)
Affinity DataIC50:  373nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237574(CHEMBL4081274)
Affinity DataIC50:  395nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237573(CHEMBL4090874)
Affinity DataIC50:  409nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237587(CHEMBL4099292)
Affinity DataIC50:  482nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50029028((cibacron blue,para isomer)1-Amino-4-{4-[4-chloro-...)
Affinity DataIC50:  625nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237576(CHEMBL4069492)
Affinity DataIC50:  746nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50029031(1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...)
Affinity DataIC50:  1.14E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268916(CHEMBL496620 | Sodium 1-Amino-4-(4-phenylthiopheny...)
Affinity DataIC50:  1.18E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336794(CHEMBL1671997 | Sodium 1-amino-4-(3-flourophenylam...)
Affinity DataIC50:  1.39E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268874(CHEMBL499580 | Sodium 1-Amino-4-[3-(4,6-dichloro-[...)
Affinity DataIC50:  1.45E+3nMAssay Description:Antagonist activity against human P2Y4 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336790(CHEMBL1671993 | Sodium 1-amino-4-(3-ethylphenylami...)
Affinity DataIC50:  1.51E+3nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237562(CHEMBL4090513)
Affinity DataIC50:  1.54E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237561(CHEMBL4082692)
Affinity DataIC50:  1.65E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237580(CHEMBL4074456)
Affinity DataIC50:  1.69E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336768(CHEMBL1671995 | sodium 1-amino-4-(3-methoxyphenyla...)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237572(CHEMBL4065831)
Affinity DataIC50:  1.76E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227016(CHEMBL401859 | Sodium 1-amino-4-(4-anilinophenylam...)
Affinity DataIC50:  1.91E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336770(CHEMBL597203 | Sodium 1-amino-4-(4-phenoxyphenylam...)
Affinity DataIC50:  1.94E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227032(CHEMBL256057 | acid blue 25 | sodium 1-amino-9,10-...)
Affinity DataIC50:  1.97E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237560(CHEMBL4060811)
Affinity DataIC50:  2.20E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  2.22E+3nMAssay Description:Antagonist activity against human P2Y4 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336787(CHEMBL445413 | sodium 1-amino-9,10-dioxo-4-(m-toly...)
Affinity DataIC50:  2.22E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227020(CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylami...)
Affinity DataIC50:  2.34E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  2.37E+3nMAssay Description:Antagonist activity at human P2Y4 receptor expressed in astrocytoma cells assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227023(1-amino-4-(4-methoxyphenyl)-2-sulfoanthraquinone |...)
Affinity DataIC50:  2.59E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336791(CHEMBL402239 | sodium 1-amino-4-(2,3-dimethylpheny...)
Affinity DataIC50:  2.63E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268768(CHEMBL522053 | sodium 1-amino-4-(2-carboxy-5-chlor...)
Affinity DataIC50:  2.76E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336788(CHEMBL404450 | sodium 1-amino-9,10-dioxo-4-(p-toly...)
Affinity DataIC50:  2.82E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237557(CHEMBL4063945)
Affinity DataIC50:  2.99E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227019(CHEMBL271673 | sodium 1-amino-4-(4-chlorophenylami...)
Affinity DataIC50:  3.03E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  3.16E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237586(CHEMBL4078095)
Affinity DataIC50:  3.21E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50378648(CHEMBL599050)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237563(CHEMBL4081964)
Affinity DataIC50:  3.37E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268878(CHEMBL495605 | Sodium 1-Amino-4-(4-benzylphenylami...)
Affinity DataIC50:  3.45E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336786(CHEMBL256864 | sodium 1-amino-9,10-dioxo-4-(o-toly...)
Affinity DataIC50:  3.49E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50371702(CHEMBL402238)
Affinity DataIC50:  3.53E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336792(CHEMBL256688 | sodium 1-amino-4-(2,4-dimethylpheny...)
Affinity DataIC50:  3.58E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  3.98E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336771(CHEMBL604158 | sodium 1-amino-4-(4-fluorophenylami...)
Affinity DataIC50:  4.04E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237582(CHEMBL4072198)
Affinity DataIC50:  4.13E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237559(CHEMBL4063599)
Affinity DataIC50:  4.98E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50029031(1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...)
Affinity DataIC50:  5.75E+3nMAssay Description:Antagonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as inhibition of UTP-induced intracellular calcium mobilization b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268685(CHEMBL524064 | sodium 1-amino-4-(2-carboxyphenylam...)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50237558(CHEMBL1671994)
Affinity DataIC50:  6.45E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336772(CHEMBL1672098 | sodium 1-amino-4-(3-bromophenylami...)
Affinity DataIC50:  6.96E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268572(CHEMBL498224 | Sodium 1-amino-4-(2-phenethylamino)...)
Affinity DataIC50:  7.18E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268574(CHEMBL498423 | Sodium 1-Amino-4-(1-naphthylamino)-...)
Affinity DataIC50:  7.42E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336793(CHEMBL1671996 | Sodium 1-amino-4-(3,5-dimethoxyphe...)
Affinity DataIC50:  9.25E+3nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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