Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50011413
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106269((2-{2-[3-(3-Methoxy-benzyl)-[1,2,4]oxadiazol-5-yl]...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi:  2.30nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106250([2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106246([1-Benzenesulfonyl-4-(2-dimethylamino-ethyl)-1H-in...)
Affinity DataKi:  3nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1F(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity against 5-hydroxytryptamine 1F receptor in CHO cells using [3H]5-HT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106246([1-Benzenesulfonyl-4-(2-dimethylamino-ethyl)-1H-in...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106248(4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tet...)
Affinity DataKi:  7.20nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106255([3-(1-Benzenesulfonyl-1H-indol-4-yl)-propyl]-dimet...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106258({2-[1-(3-Chloro-benzenesulfonyl)-5-methoxy-1H-indo...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106270({2-[5-Methoxy-1-(thiophene-2-sulfonyl)-1H-indol-3-...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093054({2-[5-Methoxy-1-(naphthalene-2-sulfonyl)-1H-indol-...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106263({2-[1-(2-Chloro-benzenesulfonyl)-5-methoxy-1H-indo...)
Affinity DataKi:  11nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  11nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106267([2-(1-Benzenesulfonyl-5-methoxy-2-methyl-1H-indol-...)
Affinity DataKi:  12nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093053({2-[1-(4-Chloro-benzenesulfonyl)-5-methoxy-1H-indo...)
Affinity DataKi:  17nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  18nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106254(1-Benzenesulfonyl-3-(2-dimethylamino-ethyl)-1H-ind...)
Affinity DataKi:  19nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106247(3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic a...)
Affinity DataKi:  20nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106250([2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  23nMAssay Description:Binding affinity against dopamine receptor D3 in HEK 293 cells using [3H]spiperone radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106261([3-(2-Dimethylamino-ethyl)-5-methoxy-indol-1-yl]-p...)
Affinity DataKi:  25nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093045({2-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-ind...)
Affinity DataKi:  26nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1F(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106252([3-(2-Dimethylamino-ethyl)-5-hydroxy-indol-1-yl]-p...)
Affinity DataKi:  29nMAssay Description:Binding affinity against 5-hydroxytryptamine 1F receptor in CHO using [3H]5-HT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  29nMAssay Description:Binding affinity for 5-hydroxytryptamine 7 receptor human cloned receptors in CHO cells using [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106256(1-Benzenesulfonyl-3-(2-dimethylamino-ethyl)-1H-ind...)
Affinity DataKi:  33nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106266(2-(1-Benzenesulfonyl-5-methoxy-1H-indol-3-yl)-ethy...)
Affinity DataKi:  40nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106257(1-Benzenesulfonyl-5-methoxy-3-(2-pyrrolidin-1-yl-e...)
Affinity DataKi:  44nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106273({2-[5-Methoxy-1-(toluene-4-sulfonyl)-1H-indol-3-yl...)
Affinity DataKi:  45nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1F(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  47nMAssay Description:Binding affinity against 5-hydroxytryptamine 1F receptor in CHO cells using [3H]5-HT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106252([3-(2-Dimethylamino-ethyl)-5-hydroxy-indol-1-yl]-p...)
Affinity DataKi:  54nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106247(3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic a...)
Affinity DataKi:  59nMAssay Description:Binding affinity against dopamine receptor D2 using [3H]spiperone radioligand in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106250([2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  62nMAssay Description:Binding affinity against dopamine receptor D2 using [3H]spiperone radioligand in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106268([2-(1-Benzenesulfonyl-5-methoxy-2,3-dihydro-1H-ind...)
Affinity DataKi:  63nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi:  65nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106246([1-Benzenesulfonyl-4-(2-dimethylamino-ethyl)-1H-in...)
Affinity DataKi:  66nMAssay Description:Binding affinity against dopamine receptor D3 in HEK 293 cells using [3H]spiperone radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi:  80nMAssay Description:Binding affinity against dopamine receptor D3 in HEK 293 cells using [3H]spiperone radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106250([2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  84nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50085972([2-(5-Methoxy-2-methyl-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  89nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106246([1-Benzenesulfonyl-4-(2-dimethylamino-ethyl)-1H-in...)
Affinity DataKi:  98nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106247(3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic a...)
Affinity DataKi:  110nMAssay Description:Binding affinity against dopamine receptor D3 in HEK 293 cells using [3H]spiperone radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106247(3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic a...)
Affinity DataKi:  130nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor of rat cortical membrane using [3H]DOB radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106260([5-Methoxy-1-(toluene-4-sulfonyl)-1,3,4,5-tetrahyd...)
Affinity DataKi:  130nMAssay Description:Binding affinity as displacement of [3H]5-HT binding to 5-hydroxytryptamine 6 receptor in HeLa cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  140nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in HeLa cells was determined using [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  170nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in HeLa cells was determined using [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50106252([3-(2-Dimethylamino-ethyl)-5-hydroxy-indol-1-yl]-p...)
Affinity DataKi:  180nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor in CHO cells using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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