Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50039202
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 3.14E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 3.15E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 3.49E+4nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 4.01E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 4.54E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 4.84E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 4.93E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 5.02E+4nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 5.13E+4nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataIC50: 2.09E+5nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair

























