Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 1154
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9410BDBM9410(N-[2-(1-benzylpiperidin-4-yl)ethyl]-N-ethyl-4-(phe...)
Affinity DataIC50: 0.300nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9409BDBM9409(N-[2-(1-benzylpiperidin-4-yl)ethyl]-N-methyl-4-(ph...)
Affinity DataIC50: 0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9411BDBM9411(CHEMBL54058 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9397BDBM9397(CHEMBL59583 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 29nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9408BDBM9408(N-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-N-phenyl-ben...)
Affinity DataIC50: 35nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9400BDBM9400(CHEMBL55968 | (2E)-but-2-enedioic acid; N-[2-(1-be...)
Affinity DataIC50: 39nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9396BDBM9396(CHEMBL56001 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 51nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9391BDBM9391(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-nitrobenzami...)
Affinity DataIC50: 55nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9399BDBM9399(CHEMBL299313 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50: 69nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9395BDBM9395(CHEMBL56706 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 85nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9392BDBM9392(CHEMBL54835 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 88nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9393BDBM9393(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-formylbenzam...)
Affinity DataIC50: 120nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9406BDBM9406(CHEMBL57696 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 130nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9413BDBM9413(CHEMBL127750 | N-methyl-N-(2-{1-[(3-methylphenyl)m...)
Affinity DataIC50: 145nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9401BDBM9401(4-{[2-(1-benzylpiperidin-4-yl)ethyl]carbamoyl}-1-o...)
Affinity DataIC50: 155nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9405BDBM9405(N-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-N-methyl-ben...)
Affinity DataIC50: 170nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9388BDBM9388(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-methylbenzam...)
Affinity DataIC50: 180nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9394BDBM9394(CHEMBL55253 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50: 180nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9390BDBM9390(N-[2-(1-benzylpiperidin-4-yl)ethyl]-3-nitrobenzami...)
Affinity DataIC50: 230nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9416BDBM9416(N-methyl-N-(2-{1-[(3-nitrophenyl)methyl]piperidin-...)
Affinity DataIC50: 370nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9423BDBM9423(N-{2-[1-(cyclohexylmethyl)piperidin-4-yl]ethyl}-N-...)
Affinity DataIC50: 410nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9387BDBM9387(N-[2-(1-benzylpiperidin-4-yl)ethyl]-3-methylbenzam...)
Affinity DataIC50: 470nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9403BDBM9403(4-(1-benzylpiperidin-4-yl)-1-phenylbutan-1-one hyd...)
Affinity DataIC50: 530nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9385BDBM9385(N-(2-(1-benzylpiperidin-4-yl)ethyl)benzamide | 1-B...)
Affinity DataIC50: 560nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9412BDBM9412(N-methyl-N-(2-{1-[(2-methylphenyl)methyl]piperidin...)
Affinity DataIC50: 770nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9398BDBM9398(CHEMBL56079 | N-[2-(1-benzylpiperidin-4-yl)ethyl]p...)
Affinity DataIC50: 800nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9389BDBM9389((2E)-but-2-enedioic acid; N-[2-(1-benzylpiperidin-...)
Affinity DataIC50: 880nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9407BDBM9407(N-benzyl-N-[2-(1-benzylpiperidin-4-yl)ethyl]benzam...)
Affinity DataIC50: 940nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9386BDBM9386(N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-methylbenzam...)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9402BDBM9402((2E)-but-2-enedioic acid; N-[2-(1-benzylpiperidin-...)
Affinity DataIC50: 1.60E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9417BDBM9417(N-methyl-N-(2-{1-[(4-nitrophenyl)methyl]piperidin-...)
Affinity DataIC50: 3.30E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9418BDBM9418(N-methyl-N-{2-[1-(2-phenylethyl)piperidin-4-yl]eth...)
Affinity DataIC50: 1.30E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9415BDBM9415(CHEMBL340382 | N-methyl-N-(2-{1-[(2-nitrophenyl)me...)
Affinity DataIC50: 1.40E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9424BDBM9424(N-{2-[1-(adamantan-1-ylmethyl)piperidin-4-yl]ethyl...)
Affinity DataIC50: 2.40E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9421BDBM9421((2E)-but-2-enedioic acid; N-methyl-N-[2-(piperidin...)
Affinity DataIC50: 2.60E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9422BDBM9422(N-{2-[1-(cyclopropylmethyl)piperidin-4-yl]ethyl}-N...)
Affinity DataIC50: 3.80E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9414BDBM9414(CHEMBL127097 | N-methyl-N-(2-{1-[(4-methylphenyl)m...)
Affinity DataIC50: 4.10E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9404BDBM9404(benzyl[2-(1-benzylpiperidin-4-yl)ethyl]amine hydro...)
Affinity DataIC50: 4.60E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9420BDBM9420(N-[2-(1-benzoylpiperidin-4-yl)ethyl]-N-methylbenza...)
Affinity DataIC50: 5.20E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Tsukuba Research Laboratories

LigandChemical structure of BindingDB Monomer ID 9419BDBM9419(N-methyl-N-(2-{1-[(2E)-3-phenylprop-2-en-1-yl]pipe...)
Affinity DataIC50: 5.40E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2006
Entry Details Article
PubMed