Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50000652
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256990BDBM50256990(CHEMBL4063580)
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256943BDBM50256943(CHEMBL4088366)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261813BDBM50261813(trans-2-(para-trifluoromethylphenyl)-cyclopropylam...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256933BDBM50256933(CHEMBL4083895)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256942BDBM50256942(CHEMBL4080504)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261917BDBM50261917(trans-2-(4-chlorophenyl)-2-fluorocyclopropanamine ...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256982BDBM50256982(CHEMBL4098523)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256941BDBM50256941(CHEMBL4079589)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256940BDBM50256940(CHEMBL4103844)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256932BDBM50256932(CHEMBL4075414)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261924BDBM50261924(trans-2-Fluoro-2-(4-methoxyphenyl)cyclopropylamine...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256978BDBM50256978(CHEMBL4061133)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261915BDBM50261915(trans-2-fluoro-2-phenylcyclopropylamin | CHEMBL455...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261970BDBM50261970(cis-(+/-)-2-Fluoro-1,2-diphenylcyclopropylamine | ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256977BDBM50256977(CHEMBL4060129)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256983BDBM50256983(CHEMBL4104945)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256981BDBM50256981(CHEMBL4083013)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256985BDBM50256985(CHEMBL4087091)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261919BDBM50261919(trans-2-fluoro-2-(4-fluorophenyl)cyclopropanamine ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261922BDBM50261922(trans-2-fluoro-2-p-tolylcyclopropanamine | CHEMBL4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256984BDBM50256984(CHEMBL4074238)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256991BDBM50256991(CHEMBL4083630)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256934BDBM50256934(CHEMBL4103002)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256979BDBM50256979(CHEMBL4069807)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256993BDBM50256993(CHEMBL4076750)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256992BDBM50256992(CHEMBL4090801)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of East Anglia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256980BDBM50256980(CHEMBL4088315)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed