Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50013864
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570409(CHEMBL4857810)
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570408(CHEMBL4873687)
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570410(CHEMBL4851152)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570410(CHEMBL4851152)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570413(CHEMBL4850259)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570411(CHEMBL4877585)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570411(CHEMBL4877585)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570401(CHEMBL4879142)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570404(CHEMBL4850583)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570396(CHEMBL4871934)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570409(CHEMBL4857810)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570397(CHEMBL4852669)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570398(CHEMBL4861626)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570413(CHEMBL4850259)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570395(CHEMBL4866915)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570396(CHEMBL4871934)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570403(CHEMBL4874651)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570397(CHEMBL4852669)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570394(CHEMBL4866548)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570406(CHEMBL4862324)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570401(CHEMBL4879142)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570400(CHEMBL4876643)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570400(CHEMBL4876643)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570408(CHEMBL4873687)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570390(CHEMBL4851106)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570392(CHEMBL4870543)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570393(CHEMBL4878394)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570402(CHEMBL4856402)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570404(CHEMBL4850583)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570402(CHEMBL4856402)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570398(CHEMBL4861626)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570388(CHEMBL4858139)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570412(CHEMBL4853766)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570394(CHEMBL4866548)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570395(CHEMBL4866915)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570405(CHEMBL4874859)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570406(CHEMBL4862324)
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570407(CHEMBL4865654)
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570399(CHEMBL4846989)
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570412(CHEMBL4853766)
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570405(CHEMBL4874859)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570390(CHEMBL4851106)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570393(CHEMBL4878394)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570386(CHEMBL4864804)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570403(CHEMBL4874651)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570407(CHEMBL4865654)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570399(CHEMBL4846989)
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide 2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570391(CHEMBL4876213)
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570392(CHEMBL4870543)
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein ADM2(Human)
University of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570389(CHEMBL4867733)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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